SCHEMBL5224792

SCHEMBL5224792

COC(=O)c1cc(NCc2ccccc2)cc(N2CCCC2=O)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSD P07339 15/20 0.56
BACE1 P56817 15/20 0.56
BACE2 Q9Y5Z0 14/20 0.56
CA1 P00915 1/20 0.52
CA2 P00918 1/20 0.52
NPC1 O15118 3/20 0.50
RAB9A P51151 3/20 0.50
MEN1 O00255 1/20 0.49
TSHR P16473 1/20 0.49
KMT2A Q03164 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
RXFP1 Q9HBX9 1/20 0.48
ALDH1A1 P00352 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48
HPGD P15428 1/20 0.48
CYP2C19 P33261 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5217472 0.91 CTSD (0.58) CTSDBACE1BACE2NPC1RAB9A
SCHEMBL5223277 0.84 NPC1 (0.56) CTSDBACE1BACE2NPC1RAB9A
SCHEMBL2524379 0.83 NPC1 (0.48) CTSDBACE1BACE2NPC1RAB9A
SCHEMBL5221058 0.82 USP2 (0.46) CTSDBACE1BACE2MEN1KMT2A
SCHEMBL5224797 0.81 MEN1 (0.44) CTSDBACE1BACE2NPC1RAB9A
SCHEMBL5220917 0.81 CTSD (0.49) CTSDBACE1BACE2MEN1KMT2A
SCHEMBL5223014 0.80 CTSD (0.48) CTSDBACE1BACE2NPC1RAB9A
SCHEMBL5222055 0.80 ALDH1A1 (0.51) CTSDBACE1BACE2MEN1KMT2A
SCHEMBL475775 0.79 MEN1 (0.56) NPC1RAB9AMEN1TSHRKMT2A
SCHEMBL5219444 0.79 MEN1 (0.56) NPC1RAB9AMEN1TSHRKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567488-B1 HYDROXYETHYLAMINE DERIVATIVES FOR THE TREATMENT OF ALZHEIMER'S DISEASE GLAXO GROUP LTD (GB) 2007-02-21 EP disclosed