SCHEMBL5225031

SCHEMBL5225031

Fc1ccc(-c2ccc(-n3ncc(CN4CCC(COc5ccccn5)CC4)c3-c3ccco3)cc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SSTR5 P35346 1/20 0.36
KCNH2 Q12809 1/20 0.36
ACHE P22303 2/20 0.35
LMNA P02545 1/20 0.35
CYP2D6 P10635 1/20 0.34
DCPS Q96C86 1/20 0.34
SMO Q99835 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5225875 0.81 CYP2D6 (0.36) CYP2D6SMO
SCHEMBL2761237 0.78 SMO (0.43) LMNASMO
SCHEMBL2761009 0.78 SMO (0.43) LMNASMO
SCHEMBL2761177 0.78 DRD4 (0.42) SMO
SCHEMBL5223970 0.77 ADORA2A (0.40) KCNH2LMNASMO
Hydrochloric Acid SCHEMBL1997589 0.77 SMO (0.42) LMNASMO
SCHEMBL5222786 0.76 GRM2 (0.38) KCNH2CYP2D6SMO
SCHEMBL2761137 0.76 SMO (0.41) LMNASMO
SCHEMBL5228002 0.75 TSHR (0.39) ACHESMO
SCHEMBL5229287 0.75 EGFR (0.40) LMNASMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed