SCHEMBL5225645

SCHEMBL5225645

COc1ccc(OC)c(OCC(O)CN2C[CH]N(CCc3ccc(Cl)cc3Cl)CC2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.48
CYP2D6 P10635 1/20 0.48
HTR7 P34969 2/20 0.46
HTR1A P08908 1/20 0.46
MAPT P10636 6/20 0.44
MAPK1 P28482 1/20 0.44
NPSR1 Q6W5P4 1/20 0.43
TDP1 Q9NUW8 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
POLB P06746 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
HTT P42858 1/20 0.42
F10 P00742 4/20 0.41
PRMT5 O14744 1/20 0.41
WDR77 Q9BQA1 1/20 0.41
TP53 P04637 1/20 0.41
ABCB1 P08183 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5224759 0.92 CYP1A2 (0.48) CYP1A2CYP2D6HTR7HTR1AMAPT
SCHEMBL5223033 0.91 MEN1 (0.47) CYP1A2CYP2D6HTR7HTR1AMAPT
SCHEMBL6256607 0.84 CYP2D6 (0.47) CYP2D6HTR7HTR1AMAPTMAPK1
SCHEMBL6186218 0.80 CACNA1G (0.52) HTR7MAPTNPSR1TDP1MEN1
SCHEMBL4865613 0.80 TSHR (0.48) CYP1A2CYP2D6HTR7HTR1AMAPT
SCHEMBL4858627 0.78 CYP2D6 (0.48) CYP1A2CYP2D6HTR7HTR1AMAPT
SCHEMBL6261178 0.75 MEN1 (0.47) CYP2D6HTR7MAPTMAPK1TDP1
SCHEMBL5228642 0.74 CYP1A2 (0.47) CYP1A2
SCHEMBL5223079 0.74 CYP2D6 (0.48) CYP2D6MAPTMAPK1TDP1MEN1
SCHEMBL5221069 0.73 MEN1 (0.49) CYP1A2CYP2D6HTR7HTR1AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1806346-A1 Substituted piperazine compounds and their use as fatty acid oxidation inhibitors CV THERAPEUTICS, INC. (US) 2007-07-11 EP disclosed