SCHEMBL5223033

SCHEMBL5223033

COc1ccccc1OCC(O)CN1C[CH]N(CCc2ccc(Cl)cc2Cl)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
USP2 O75604 1/20 0.47
HTT P42858 1/20 0.47
CYP2D6 P10635 2/20 0.47
CYP1A2 P05177 1/20 0.47
MAPT P10636 5/20 0.46
HRH1 P35367 3/20 0.46
LMNA P02545 3/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 2/20 0.44
HTR1A P08908 1/20 0.44
HTR7 P34969 1/20 0.44
F8 P00451 1/20 0.43
F5 P12259 1/20 0.43
TP53 P04637 1/20 0.43
CYP3A4 P08684 1/20 0.42
TSHR P16473 1/20 0.42
NFKB1 P19838 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5225645 0.91 CYP1A2 (0.48) MEN1KMT2AHTTCYP2D6CYP1A2
SCHEMBL5224759 0.83 CYP1A2 (0.48) MEN1KMT2AHTTCYP2D6CYP1A2
SCHEMBL5221069 0.80 MEN1 (0.49) MEN1KMT2AUSP2HTTCYP2D6
SCHEMBL6256607 0.80 CYP2D6 (0.47) MEN1KMT2AHTTCYP2D6MAPT
SCHEMBL4861739 0.79 CYP2D6 (0.58) MEN1KMT2AUSP2HTTCYP2D6
SCHEMBL5228642 0.76 CYP1A2 (0.47) CYP1A2CYP3A4
SCHEMBL2332160 0.74 LMNA (0.73) MEN1KMT2AUSP2HTTCYP2D6
SCHEMBL6184593 0.73 HRH1 (0.46) MEN1KMT2AUSP2HTTCYP2D6
SCHEMBL4865613 0.71 TSHR (0.48) MEN1KMT2AUSP2CYP2D6CYP1A2
SCHEMBL6186218 0.71 CACNA1G (0.52) MEN1KMT2AHTTMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1806346-A1 Substituted piperazine compounds and their use as fatty acid oxidation inhibitors CV THERAPEUTICS, INC. (US) 2007-07-11 EP disclosed