SCHEMBL5225949

SCHEMBL5225949

Cn1c(N(C(=O)O)c2ccccc2)nc2cc([N+](=O)[O-])ccc21

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.49
LMNA P02545 5/20 0.49
KMT2A Q03164 5/20 0.49
MAPT P10636 2/20 0.49
KDM4E B2RXH2 1/20 0.49
APOBEC3A P31941 1/20 0.49
HTT P42858 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
APOBEC3G Q9HC16 1/20 0.49
PKM P14618 4/20 0.47
SMN1; SMN2 Q16637 1/20 0.46
CYP19A1 P11511 1/20 0.45
HDAC6 Q9UBN7 2/20 0.45
RAB9A P51151 2/20 0.44
NPC1 O15118 1/20 0.44
MEN1 O00255 2/20 0.44
CYP2D6 P10635 1/20 0.44
RXFP1 Q9HBX9 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5225943 1.00 ALDH1A1 (0.49) ALDH1A1LMNAKMT2AMAPTKDM4E
SCHEMBL5229039 0.91 KMT2A (0.44) ALDH1A1LMNAKMT2AMAPTKDM4E
SCHEMBL5229049 0.91 KMT2A (0.44) ALDH1A1LMNAKMT2AMAPTKDM4E
SCHEMBL5226510 0.88 MAPT (0.54) ALDH1A1LMNAKMT2AMAPTKDM4E
SCHEMBL4976760 0.86 ALDH1A1 (0.44) ALDH1A1LMNAKMT2AMAPTKDM4E
SCHEMBL5223908 0.84 ALDH1A1 (0.44) ALDH1A1LMNAKMT2AMAPTKDM4E
SCHEMBL5226357 0.81 HDAC6 (0.48) ALDH1A1MAPTKDM4EHTTPKM
SCHEMBL4978503 0.77 KMT2A (0.42) ALDH1A1LMNAKMT2AMAPTKDM4E
SCHEMBL4978681 0.76 MAPT (0.41) ALDH1A1LMNAKMT2AMAPTKDM4E
SCHEMBL4978620 0.75 MAPT (0.50) ALDH1A1LMNAKMT2AMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1487824-B1 DIAMINO-PYRIMIDINES AND THEIR USE AS ANGIOGENESIS INHIBITORS SMITHKLINE BEECHAM CORP (US) 2007-06-20 EP disclosed