SCHEMBL5226008

SCHEMBL5226008

CC(C)COC(=O)N1CCC(CC2CCN(C)CC2)CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 1/20 0.44
GAA P10253 1/20 0.40
NOS3 P29474 1/20 0.38
NOS2 P35228 1/20 0.38
GPR119 Q8TDV5 2/20 0.38
L3MBTL1 Q9Y468 2/20 0.37
THRB P10828 1/20 0.37
ATM Q13315 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37
CHRM2 P08172 1/20 0.37
CHRM1 P11229 1/20 0.37
HSD11B1 P28845 1/20 0.37
KIT P10721 1/20 0.37
GNAI3 P08754 1/20 0.37
GNAO1 P09471 1/20 0.37
GNAI1 P63096 1/20 0.37
HRH2 P25021 1/20 0.36
HRH1 P35367 1/20 0.36
DRD2 P14416 1/20 0.36
PRMT5 O14744 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5219039 0.87 RAB9A (0.43) RAB9AGAANOS3NOS2GPR119
SCHEMBL5217684 0.85 RAB9A (0.43) RAB9AGAANOS3NOS2GPR119
SCHEMBL5221871 0.85 RAB9A (0.43) RAB9AGAANOS3NOS2GPR119
SCHEMBL5221770 0.84 RAB9A (0.42) RAB9AGAANOS3NOS2GPR119
SCHEMBL5225927 0.83 CHRM1 (0.46) RAB9AGAAL3MBTL1THRBATM
SCHEMBL1693216 0.83 RAB9A (0.48) RAB9AGAANOS3NOS2GPR119
SCHEMBL10089204 0.83 RAB9A (0.48) RAB9AGAANOS3NOS2GPR119
SCHEMBL4977215 0.83 RAB9A (0.48) RAB9AGAANOS3NOS2GPR119
SCHEMBL8921640 0.82 RAB9A (0.45) RAB9AHRH3KITHRH2HRH1
SCHEMBL2894884 0.81 TPSAB1 (0.47) RAB9AGAANOS3NOS2GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1789410-A1 METHYLENE DIPIPERIDINE DERIVATIVES GLAXO GROUP LIMITED (GB) 2007-05-30 EP disclosed
WO-2006029906-A1 METHYLENE DIPIPERIDINE DERIVATIVES GLAXO GROUP LIMITED (GB) 2006-03-23 WO disclosed