SCHEMBL5226484

SCHEMBL5226484

COc1ccc(-c2ccc(-n3ncc(CN4CCN(C5CCCC5)CC4)c3-c3ccco3)cc2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMO Q99835 2/20 0.45
MAPT P10636 3/20 0.43
DRD4 P21917 1/20 0.41
DRD3 P35462 1/20 0.41
NPBWR1 P48145 1/20 0.40
MCHR1 Q99705 1/20 0.40
TP53 P04637 2/20 0.39
KDM4E B2RXH2 2/20 0.39
HRH3 Q9Y5N1 1/20 0.39
ALDH1A1 P00352 2/20 0.38
ACHE P22303 1/20 0.38
TSHR P16473 2/20 0.38
HPGD P15428 1/20 0.38
HSD17B10 Q99714 1/20 0.38
PTGS1 P23219 1/20 0.38
PTGS2 P35354 1/20 0.38
P2RX3 P56373 1/20 0.37
LMNA P02545 1/20 0.36
TLR9 Q9NR96 1/20 0.36
TLR7 Q9NYK1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2761177 0.88 DRD4 (0.42) SMOMAPTDRD4DRD3TP53
SCHEMBL5224302 0.87 SMO (0.49) SMOMAPTNPBWR1MCHR1TP53
SCHEMBL5232263 0.87 SMO (0.49) SMOMAPTNPBWR1MCHR1TP53
SCHEMBL5226663 0.84 KMT2A (0.44) DRD4DRD3TP53KDM4EALDH1A1
SCHEMBL5226986 0.84 DRD4 (0.39) SMOMAPTDRD4DRD3MCHR1
SCHEMBL5230456 0.84 SMO (0.46) SMOMAPTNPBWR1MCHR1TP53
SCHEMBL5225260 0.84 KMT2A (0.39) DRD4DRD3TP53KDM4EALDH1A1
SCHEMBL5228505 0.83 F10 (0.48)
SCHEMBL5226667 0.80 DRD4 (0.39) SMODRD4DRD3KDM4EHRH3
SCHEMBL2761078 0.78 DRD4 (0.40) MAPTDRD4DRD3TP53KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed