SCHEMBL5232263

SCHEMBL5232263

COc1ccc(-c2ccc(-n3ncc(CN4CCN(C)CC4)c3-c3ccco3)cc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMO Q99835 2/20 0.49
CHKA P35790 1/20 0.44
NPBWR1 P48145 1/20 0.43
MCHR1 Q99705 1/20 0.43
PTGS1 P23219 1/20 0.41
PTGS2 P35354 1/20 0.41
KDM4E B2RXH2 3/20 0.40
TP53 P04637 2/20 0.40
KDM5B Q9UGL1 1/20 0.40
MAPT P10636 3/20 0.39
ALDH1A1 P00352 4/20 0.39
LMNA P02545 4/20 0.39
TSHR P16473 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39
MAP3K11 Q16584 1/20 0.38
MAPK1 P28482 1/20 0.38
NTSR1 P30989 1/20 0.38
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5224302 0.92 SMO (0.49) SMONPBWR1MCHR1PTGS1PTGS2
SCHEMBL5230456 0.89 SMO (0.46) SMONPBWR1MCHR1PTGS1PTGS2
SCHEMBL2761009 0.88 SMO (0.43) SMOCHKAPTGS1TP53MAPT
SCHEMBL5226484 0.87 SMO (0.45) SMONPBWR1MCHR1PTGS1PTGS2
SCHEMBL5228505 0.84 F10 (0.48)
SCHEMBL5224673 0.84 SMO (0.40) SMOKDM4EALDH1A1LMNA
SCHEMBL5222920 0.84 ALDH1A1 (0.41) KDM4ETP53MAPTALDH1A1LMNA
SCHEMBL5230509 0.83 POLB (0.41) SMOKDM4ETP53ALDH1A1TSHR
SCHEMBL5228457 0.83 PIK3R1 (0.39) SMOCHKAMAPTALDH1A1
SCHEMBL5228410 0.82 PTGS1 (0.49) NPBWR1MCHR1PTGS1PTGS2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed