SCHEMBL5226986

SCHEMBL5226986

Fc1cccc(-c2ccc(-n3ncc(CN4CCN(C5CCCC5)CC4)c3-c3ccco3)cc2)c1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 1/20 0.39
DRD3 P35462 1/20 0.39
POLB P06746 1/20 0.39
KDM2B Q8NHM5 1/20 0.38
ALDH1A1 P00352 2/20 0.37
SIGMAR1 Q99720 1/20 0.36
SMO Q99835 1/20 0.35
TP53 P04637 1/20 0.35
MAPT P10636 1/20 0.35
MCHR1 Q99705 1/20 0.35
ALPL P05186 1/20 0.34
CXCR3 P49682 1/20 0.34
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
GAA P10253 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2761177 0.92 DRD4 (0.42) DRD4DRD3POLBALDH1A1SMO
SCHEMBL5229287 0.87 EGFR (0.40) ALDH1A1SMOALPLCXCR3KDM4E
SCHEMBL5226613 0.87 SMO (0.40) DRD4DRD3POLBALDH1A1SMO
SCHEMBL5224673 0.87 SMO (0.40) DRD4DRD3ALDH1A1SMOALPL
SCHEMBL5226663 0.86 KMT2A (0.44) DRD4DRD3POLBALDH1A1TP53
SCHEMBL5225260 0.86 KMT2A (0.39) DRD4DRD3POLBALDH1A1TP53
SCHEMBL5224744 0.85 HTR1A (0.38) ALDH1A1SMOALPLKDM4ELMNA
SCHEMBL5226484 0.84 SMO (0.45) DRD4DRD3ALDH1A1SMOTP53
SCHEMBL2761078 0.84 DRD4 (0.40) DRD4DRD3POLBALDH1A1TP53
SCHEMBL5228047 0.84 HTR2C (0.37) DRD4ALDH1A1MCHR1ALPLCXCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed