SCHEMBL5226667

SCHEMBL5226667

c1ccc(CC2=C(c3ccc(-n4ncc(CN5CCN(C6CCCC6)CC5)c4-c4ccco4)cc3)OCO2)cc1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 2/20 0.39
DRD3 P35462 2/20 0.39
TSHR P16473 2/20 0.35
TRPV6 Q9H1D0 4/20 0.35
ALDH1A1 P00352 3/20 0.35
KDM4E B2RXH2 4/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
HRH3 Q9Y5N1 1/20 0.34
DRD2 P14416 2/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
SMO Q99835 1/20 0.34
HTR2A P28223 1/20 0.34
HRH1 P35367 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.33
HCRTR1 O43613 1/20 0.33
HTR1D P28221 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5229345 0.88 EGFR (0.34) DRD4DRD3TSHRALDH1A1KDM4E
SCHEMBL5222928 0.88 SMO (0.38) DRD4DRD3ALDH1A1KDM4ESMN1; SMN2
SCHEMBL5226173 0.88 SMO (0.38) DRD4DRD3ALDH1A1KDM4ESMN1; SMN2
SCHEMBL5226844 0.86 SIGMAR1 (0.34) DRD4DRD3ALDH1A1KDM4ESMN1; SMN2
SCHEMBL5226450 0.85 F10 (0.35) ALDH1A1KMT2A
SCHEMBL5225471 0.83 HRH3 (0.35) DRD4DRD3KDM4EHRH3DRD2
SCHEMBL2761177 0.82 DRD4 (0.42) DRD4DRD3TSHRTRPV6ALDH1A1
SCHEMBL5226663 0.81 KMT2A (0.44) DRD4DRD3TSHRTRPV6ALDH1A1
SCHEMBL5230408 0.81 SLC2A1 (0.32) TSHRALDH1A1SMN1; SMN2L3MBTL1HCRTR1
SCHEMBL5226484 0.80 SMO (0.45) DRD4DRD3TSHRALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed