SCHEMBL5226589

SCHEMBL5226589

COc1ccc(-c2nc3cc(OC)ccc3o2)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.68
RAB9A P51151 6/20 0.68
ALDH1A1 P00352 4/20 0.68
MAPT P10636 4/20 0.68
HDAC6 Q9UBN7 2/20 0.65
THRB P10828 1/20 0.62
UTRN P46939 1/20 0.62
SMN1; SMN2 Q16637 5/20 0.61
HSD17B10 Q99714 4/20 0.61
TP53 P04637 4/20 0.61
HPGD P15428 3/20 0.61
L3MBTL1 Q9Y468 3/20 0.61
NFKB1 P19838 2/20 0.61
NFKB2 Q00653 2/20 0.61
RELA Q04206 2/20 0.61
KDM4E B2RXH2 2/20 0.61
TDP1 Q9NUW8 2/20 0.61
GLA P06280 1/20 0.61
PTPN2 P17706 3/20 0.61
PTPN1 P18031 3/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12639220 0.93 NPC1 (0.68) NPC1RAB9AALDH1A1MAPTHDAC6
SCHEMBL11828034 0.92 ALDH1A1 (0.71) NPC1RAB9AALDH1A1MAPTHDAC6
SCHEMBL5413693 0.91 ESR1 (0.69) NPC1RAB9AALDH1A1MAPTHDAC6
SCHEMBL18726342 0.91 RAB9A (0.69) NPC1RAB9AALDH1A1MAPTHDAC6
SCHEMBL4032178 0.91 MAPT (0.60) NPC1RAB9AALDH1A1MAPTHDAC6
SCHEMBL28559369 0.90 SMN1; SMN2 (0.66) NPC1RAB9AALDH1A1MAPTHDAC6
SCHEMBL11138585 0.90 HDAC6 (0.58) NPC1RAB9AALDH1A1MAPTHDAC6
SCHEMBL9858278 0.90 HDAC6 (0.58) NPC1RAB9AALDH1A1MAPTHDAC6
SCHEMBL1024034 0.89 HSD17B10 (0.78) NPC1RAB9AALDH1A1MAPTHDAC6
SCHEMBL2246136 0.89 ALDH1A1 (0.78) NPC1RAB9AALDH1A1MAPTHDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1781628-A2 PRODRUG SUBSTITUTED BENZOXAZOLES AS ESTROGENIC AGENTS Wyeth a Corporation of the State of Delaware (US) 2007-05-09 EP disclosed
WO-2006026316-A2 PRODRUG SUBSTITUTED BENZOXAZOLES AS ESTROGENIC AGENTS WYETH (US) 2006-03-09 WO disclosed