SCHEMBL5228082

SCHEMBL5228082

NC[C@H](O)C1CCCCC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 1.00
KDM4E B2RXH2 2/20 0.95
GMNN O75496 1/20 0.95
LMNA P02545 1/20 0.95
MAPT P10636 1/20 0.95
BLM P54132 1/20 0.95
PMP22 Q01453 1/20 0.95
SMN1; SMN2 Q16637 1/20 0.95
EPHX1 P07099 2/20 0.56
ALDH1A1 P00352 1/20 0.47
SHBG P04278 1/20 0.39
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
SLC6A3 Q01959 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL133228 1.00 TP53 (1.00) TP53KDM4EGMNNLMNAMAPT
SCHEMBL4078170 1.00 TP53 (1.00) TP53KDM4EGMNNLMNAMAPT
SCHEMBL23270700 1.00 TP53 (1.00) TP53KDM4EGMNNLMNAMAPT
SCHEMBL4079339 1.00 TP53 (1.00) TP53KDM4EGMNNLMNAMAPT
Hydrochloric Acid SCHEMBL160732 0.97 KDM4E (1.00) TP53KDM4EGMNNLMNAMAPT
Hydrochloric Acid SCHEMBL2063394 0.97 KDM4E (1.00) TP53KDM4EGMNNLMNAMAPT
SCHEMBL3647508 0.97
SCHEMBL22535894 0.97
Hydrochloric Acid SCHEMBL19642704 0.95 KDM4E (0.95) TP53KDM4EGMNNLMNAMAPT
Hydrochloric Acid SCHEMBL30187467 0.95 KDM4E (0.95) TP53KDM4EGMNNLMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12291535-B2 Benzodiazepine derivatives, compositions, and methods for treating cognitive impairment AGENEBIO, INC. (US) 2025-05-06 US disclosed
CN-112601749-B Benzodiazepine derivatives, compositions and methods for treating cognitive impairment 艾吉因生物股份有限公司 2024-03-26 CN disclosed
US-20230107032-A1 BENZODIAZEPINE DERIVATIVES, COMPOSITIONS, AND METHODS FOR TREATING COGNITIVE IMPAIRMENT NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2023-04-06 US disclosed
US-11414425-B2 Benzodiazepine derivatives, compositions, and methods for treating cognitive impairment AGENEBIO, INC. (US) 2022-08-16 US disclosed
EP-3168208-A1 PROCESSES FOR THE PREPARATION OF DIASTEREOMERICALLY AND ENANTIOMERICALLY ENRICHED OXAZOLINES Quimica Sintetica, S.A. (ES) 2017-05-17 EP disclosed
EP-1765817-A1 THIAZOLINONE UNSUBSTITUTED QUINOLINES F.HOFFMANN-LA ROCHE AG (CH) 2007-03-28 EP disclosed
WO-2006002829-A1 THIAZOLINONE UNSUBSTITUTED QUINOLINES F. HOFFMANN-LA ROCHE AG (CH) 2006-01-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230107032-A1 BENZODIAZEPINE DERIVATIVES, COMPOSITIONS, AND METHODS FOR TREATING COGNITIVE IMPAIRMENT GABRA5, GRM5, GABRA1 TP53 443/4885KDM4E 2690/4885GMNN 4334/4885
US-11414425-B2 Benzodiazepine derivatives, compositions, and methods for treating cognitive impairment GABRA5, GRM5, GABRA1 TP53 443/4885KDM4E 2690/4885GMNN 4334/4885
US-12291535-B2 Benzodiazepine derivatives, compositions, and methods for treating cognitive impairment GABRA5, GRM5, GABRA1 TP53 443/4885KDM4E 2690/4885GMNN 4334/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.