SCHEMBL5228219

SCHEMBL5228219

CN1CCN(Cc2cnn(-c3ccc(-c4ccc(F)cc4)cc3)c2-c2c(F)cccc2F)CC1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SMO Q99835 2/20 0.47
MAP4K1 Q92918 5/20 0.45
DRD4 P21917 4/20 0.42
DRD3 P35462 4/20 0.42
DRD2 P14416 3/20 0.42
MAPK14 Q16539 2/20 0.41
MAPT P10636 2/20 0.41
MC4R P32245 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
ALDH1A1 P00352 1/20 0.39
TNIK Q9UKE5 1/20 0.38
HTR6 P50406 1/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2761123 0.90 SMO (0.50) SMOMAP4K1DRD4MAPTL3MBTL1
SCHEMBL5737789 0.88 SMO (0.44) SMODRD4DRD3DRD2MAPK14
SCHEMBL5228124 0.83 SMO (0.43) SMODRD4DRD3DRD2MAPK14
SCHEMBL5230174 0.83 DRD4 (0.46) SMODRD4DRD3DRD2MAPK14
SCHEMBL1689504 0.83 SMO (0.45) SMOMAP4K1DRD4DRD3DRD2
SCHEMBL5224153 0.83 BRD4 (0.44) SMODRD4DRD3DRD2MAPT
SCHEMBL2761009 0.82 SMO (0.43) SMODRD4DRD3DRD2MAPK14
SCHEMBL5226797 0.82 SMO (0.61) SMOMAPK14MAPTL3MBTL1ALDH1A1
SCHEMBL2761085 0.82 DHODH (0.43) SMOMAP4K1DRD4DRD3DRD2
SCHEMBL5226795 0.82 SMO (0.42) SMODRD4DRD3DRD2MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed