SCHEMBL5230174

SCHEMBL5230174

CN1CCN(Cc2cnn(-c3ccc(-c4ccc(F)cc4)cc3)c2-c2cccc(Cl)c2)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 3/20 0.46
DRD3 P35462 3/20 0.46
DRD2 P14416 2/20 0.46
SMO Q99835 1/20 0.46
ALDH1A1 P00352 4/20 0.42
MAPT P10636 3/20 0.42
MAPK14 Q16539 1/20 0.41
AXL P30530 1/20 0.40
TNIK Q9UKE5 1/20 0.40
HTR6 P50406 1/20 0.40
KDM4E B2RXH2 3/20 0.39
PKM P14618 1/20 0.39
TP53 P04637 1/20 0.39
ALPI P09923 1/20 0.39
ALPG P10696 1/20 0.39
FNTA P49354 1/20 0.39
PGGT1B P53609 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
POLB P06746 1/20 0.38
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5227445 0.92 DRD4 (0.46) DRD4DRD3DRD2SMOALDH1A1
SCHEMBL5230607 0.91 DRD4 (0.46) DRD4DRD3DRD2SMOALDH1A1
SCHEMBL5227774 0.90 DRD3 (0.45) DRD4DRD3DRD2SMOALDH1A1
SCHEMBL5229642 0.87 DRD2 (0.42) DRD4DRD3DRD2SMOMAPT
SCHEMBL5226797 0.86 SMO (0.61) SMOALDH1A1MAPTMAPK14HTR6
SCHEMBL5226907 0.86 DRD4 (0.43) DRD4DRD3DRD2SMOALDH1A1
SCHEMBL5228219 0.83 SMO (0.47) DRD4DRD3DRD2SMOALDH1A1
SCHEMBL5228024 0.83 HTR2C (0.42) DRD4DRD3DRD2SMOTP53
SCHEMBL5228124 0.82 SMO (0.43) DRD4DRD3DRD2SMOMAPT
SCHEMBL5226795 0.81 SMO (0.42) DRD4DRD3DRD2SMOALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed