SCHEMBL5228638

SCHEMBL5228638

CN1CCN(Cc2cnn(-c3ccc(-c4ccncc4)cc3)c2-c2ccccc2F)CC1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 2/20 0.41
DRD3 P35462 2/20 0.41
SMO Q99835 3/20 0.40
DRD2 P14416 1/20 0.40
SSTR5 P35346 1/20 0.38
MELK Q14680 2/20 0.38
ALDH1A1 P00352 2/20 0.37
STAT1 P42224 1/20 0.37
HTT P42858 1/20 0.37
MAP4K1 Q92918 2/20 0.37
MAPK14 Q16539 2/20 0.37
TGFBR1 P36897 1/20 0.36
ACHE P22303 1/20 0.36
BMP4 P12644 1/20 0.36
MAPT P10636 1/20 0.36
CSNK1D P48730 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1689504 0.93 SMO (0.45) DRD4DRD3SMODRD2SSTR5
SCHEMBL5737789 0.92 SMO (0.44) DRD4DRD3SMODRD2SSTR5
SCHEMBL7256544 0.92 DRD4 (0.44) DRD4DRD3SMODRD2SSTR5
SCHEMBL5232121 0.89 DRD4 (0.39) DRD4DRD3SMODRD2SSTR5
SCHEMBL7261049 0.89 CHKA (0.50) DRD4DRD3SMODRD2SSTR5
SCHEMBL5227503 0.88 DRD4 (0.42) DRD4DRD3SMODRD2SSTR5
SCHEMBL2761085 0.87 DHODH (0.43) DRD4DRD3SMODRD2SSTR5
SCHEMBL5225912 0.87 MAP4K1 (0.41) DRD4DRD3SMODRD2SSTR5
SCHEMBL5224217 0.87 SMO (0.44) DRD4DRD3SMODRD2SSTR5
SCHEMBL7261173 0.87 SMO (0.47) DRD4DRD3SMODRD2SSTR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed