SCHEMBL5227503

SCHEMBL5227503

CN1CCN(Cc2cnn(-c3ccc(-c4ccc(N(C)C)cc4)cc3)c2-c2ccccc2F)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 2/20 0.42
DRD3 P35462 2/20 0.42
SMO Q99835 3/20 0.39
DRD2 P14416 1/20 0.39
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
SSTR5 P35346 1/20 0.37
MAP4K1 Q92918 3/20 0.36
ALDH1A1 P00352 3/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2D6 P10635 2/20 0.36
MAPK1 P28482 2/20 0.36
HSD17B10 Q99714 2/20 0.36
MAPT P10636 2/20 0.36
KDM4E B2RXH2 1/20 0.36
TP53 P04637 1/20 0.36
HPGD P15428 1/20 0.36
TSHR P16473 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1689504 0.91 SMO (0.45) DRD4DRD3SMODRD2SSTR5
SCHEMBL5737789 0.90 SMO (0.44) DRD4DRD3SMODRD2SSTR5
SCHEMBL7256544 0.90 DRD4 (0.44) DRD4DRD3SMODRD2SSTR5
SCHEMBL5228638 0.88 DRD4 (0.41) DRD4DRD3SMODRD2SSTR5
SCHEMBL7261049 0.87 CHKA (0.50) DRD4DRD3SMODRD2SSTR5
SCHEMBL2761085 0.85 DHODH (0.43) DRD4DRD3SMODRD2SSTR5
SCHEMBL5225912 0.85 MAP4K1 (0.41) DRD4DRD3SMODRD2SSTR5
SCHEMBL5232121 0.85 DRD4 (0.39) DRD4DRD3SMODRD2SSTR5
SCHEMBL5224217 0.85 SMO (0.44) DRD4DRD3SMODRD2NPC1
SCHEMBL5230137 0.85 PTGS2 (0.43) DRD4DRD3SMODRD2SSTR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed