SCHEMBL5224217

SCHEMBL5224217

CN1CCN(Cc2cnn(-c3ccc(-c4ccc(Oc5ccccc5)cc4)cc3)c2-c2ccccc2F)CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMO Q99835 4/20 0.44
DRD4 P21917 2/20 0.40
DRD3 P35462 2/20 0.40
DRD2 P14416 1/20 0.40
MAP4K1 Q92918 1/20 0.40
SSTR5 P35346 1/20 0.39
TRPV4 Q9HBA0 1/20 0.38
ACHE P22303 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
ALDH1A1 P00352 1/20 0.38
TNK2 Q07912 1/20 0.37
SCN9A Q15858 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
CXCR1 P25024 1/20 0.37
LMNA P02545 1/20 0.36
GAA P10253 1/20 0.36
ALK Q9UM73 1/20 0.36
KDM5B Q9UGL1 1/20 0.36
ADORA2A P29274 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1689504 0.92 SMO (0.45) SMODRD4DRD3DRD2MAP4K1
SCHEMBL5737789 0.89 SMO (0.44) SMODRD4DRD3DRD2SSTR5
SCHEMBL7256544 0.89 DRD4 (0.44) SMODRD4DRD3DRD2MAP4K1
SCHEMBL7261049 0.88 CHKA (0.50) SMODRD4DRD3DRD2SSTR5
SCHEMBL5228638 0.87 DRD4 (0.41) SMODRD4DRD3DRD2MAP4K1
SCHEMBL5227503 0.85 DRD4 (0.42) SMODRD4DRD3DRD2MAP4K1
SCHEMBL7261888 0.85 ALDH1A1 (0.49) SMODRD4DRD3DRD2SSTR5
SCHEMBL5232121 0.85 DRD4 (0.39) SMODRD4DRD3DRD2MAP4K1
SCHEMBL2761085 0.85 DHODH (0.43) SMODRD4DRD3DRD2MAP4K1
SCHEMBL5225912 0.85 MAP4K1 (0.41) SMODRD4DRD3DRD2MAP4K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed