SCHEMBL5232121

SCHEMBL5232121

CN1CCN(Cc2cnn(-c3ccc(-c4ccsc4)cc3)c2-c2ccccc2F)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 3/20 0.39
DRD3 P35462 3/20 0.39
SMO Q99835 3/20 0.38
DRD2 P14416 2/20 0.38
KDR P35968 3/20 0.37
FLT1 P17948 2/20 0.37
FLT4 P35916 2/20 0.37
STAT1 P42224 1/20 0.37
HTT P42858 1/20 0.37
SSTR5 P35346 1/20 0.37
GABRG2 P18507 1/20 0.36
GABRB3 P28472 1/20 0.36
GABRA3 P34903 1/20 0.36
ALDH1A1 P00352 3/20 0.36
MAP4K1 Q92918 2/20 0.35
KIT P10721 1/20 0.35
TEK Q02763 1/20 0.35
ACHE P22303 1/20 0.35
MAPT P10636 1/20 0.35
MEN1 O00255 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1689504 0.90 SMO (0.45) DRD4DRD3SMODRD2KDR
SCHEMBL5738329 0.90 CYP2A13 (0.43) DRD4DRD3SMODRD2KDR
SCHEMBL5228638 0.89 DRD4 (0.41) DRD4DRD3SMODRD2STAT1
SCHEMBL5737789 0.89 SMO (0.44) DRD4DRD3SMODRD2SSTR5
SCHEMBL7256544 0.89 DRD4 (0.44) DRD4DRD3SMODRD2SSTR5
SCHEMBL5226383 0.87 DRD3 (0.44) DRD4DRD3SMODRD2KDR
SCHEMBL7261049 0.86 CHKA (0.50) DRD4DRD3SMODRD2KDR
SCHEMBL5227503 0.85 DRD4 (0.42) DRD4DRD3SMODRD2KDR
SCHEMBL5226795 0.85 SMO (0.42) DRD4DRD3SMODRD2KDR
SCHEMBL5224217 0.85 SMO (0.44) DRD4DRD3SMODRD2SSTR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed
WO-2003031435-A1 PYRAZOLE DERIVATIVES AS GLYCINE TRANSPORTER INHIBITORS MERCK PATENT GMBH (DE) 2003-04-17 WO disclosed