SCHEMBL5228692

SCHEMBL5228692

Fc1ccc(-c2ccc(-n3ncc(CNCCc4ccccn4)c3-c3ccco3)cc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.47
CYP2D6 P10635 1/20 0.47
KDM4E B2RXH2 3/20 0.45
LMNA P02545 3/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.39
ALDH1A1 P00352 3/20 0.38
GFER P55789 1/20 0.38
TGFBR1 P36897 1/20 0.37
TGFBR2 P37173 1/20 0.37
FLT3 P36888 1/20 0.36
DPP7 Q9UHL4 1/20 0.36
HTT P42858 1/20 0.35
GRIN1 Q05586 1/20 0.35
GRIN2B Q13224 1/20 0.35
PTGS1 P23219 1/20 0.34
GAA P10253 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5226789 0.85 ALDH1A1 (0.39) CYP2D6KDM4ELMNAMEN1KMT2A
SCHEMBL5231186 0.82 SMN1; SMN2 (0.38) CYP1A2CYP2D6KDM4ELMNAMEN1
SCHEMBL5224886 0.82 PTGS1 (0.37) CYP2D6KDM4ELMNAMEN1KMT2A
SCHEMBL5228534 0.81 PTGS1 (0.36) CYP2D6KDM4ELMNAMEN1KMT2A
SCHEMBL5224632 0.81 ALDH1A1 (0.39) CYP2D6KDM4ELMNAMEN1KMT2A
SCHEMBL5230237 0.80 MAPT (0.47) KDM4EMEN1KMT2ARAB9ASMN1; SMN2
SCHEMBL5227606 0.80 TP53 (0.42) CYP2D6LMNASMN1; SMN2ALDH1A1PTGS1
SCHEMBL5228370 0.79 ALDH1A1 (0.36) CYP2D6KDM4ELMNARAB9ASMN1; SMN2
SCHEMBL5226111 0.78 CHRM2 (0.36) CYP1A2CYP2D6KDM4ELMNAKMT2A
SCHEMBL5223225 0.77 PTGS1 (0.36) CYP2D6KDM4ELMNASMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed