SCHEMBL5230237

SCHEMBL5230237

COc1ccc(-c2ccc(-n3ncc(CNCc4ccccn4)c3-c3ccco3)cc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.47
KDM4E B2RXH2 5/20 0.47
ALDH1A1 P00352 4/20 0.47
HPGD P15428 3/20 0.47
HSD17B10 Q99714 3/20 0.47
RAB9A P51151 3/20 0.47
NPC1 O15118 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
NPBWR1 P48145 2/20 0.41
MCHR1 Q99705 1/20 0.41
TP53 P04637 4/20 0.41
GSK3B P49841 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
PTGS1 P23219 1/20 0.39
PTGS2 P35354 1/20 0.39
ALPL P05186 1/20 0.39
ALPG P10696 1/20 0.39
TSHR P16473 1/20 0.39
MAPK1 P28482 1/20 0.39
MEN1 O00255 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5225666 0.82 NPBWR1 (0.43) MAPTKDM4EALDH1A1HPGDHSD17B10
SCHEMBL5228692 0.80 CYP1A2 (0.47) MAPTKDM4EALDH1A1HPGDHSD17B10
SCHEMBL5230220 0.79 NPBWR1 (0.40) MAPTKDM4EALDH1A1HPGDHSD17B10
SCHEMBL5228410 0.79 PTGS1 (0.49) MAPTKDM4EALDH1A1HPGDHSD17B10
SCHEMBL5226619 0.78 NPBWR1 (0.47) MAPTKDM4EALDH1A1HPGDHSD17B10
SCHEMBL5224717 0.76 NPBWR1 (0.45) MAPTKDM4EALDH1A1HPGDHSD17B10
SCHEMBL5232263 0.74 SMO (0.49) MAPTKDM4EALDH1A1HPGDHSD17B10
SCHEMBL5224302 0.74 SMO (0.49) MAPTKDM4EALDH1A1HPGDHSD17B10
SCHEMBL5229004 0.73 NPBWR1 (0.40) MAPTKDM4EALDH1A1HPGDHSD17B10
SCHEMBL5230456 0.73 SMO (0.46) MAPTKDM4EALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed