SCHEMBL5229799

SCHEMBL5229799

COc1ccc2c(c1)=COCC=2

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 3/20 0.36
CA1 P00915 3/20 0.36
CA7 P43166 3/20 0.36
CA9 Q16790 3/20 0.36
CA14 Q9ULX7 3/20 0.36
CA2 P00918 2/20 0.36
CYP1A2 P05177 2/20 0.35
CYP2A6 P11509 1/20 0.35
DRD2 P14416 2/20 0.35
DRD3 P35462 2/20 0.35
DRD1 P21728 1/20 0.35
DRD5 P21918 1/20 0.35
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
POLB P06746 1/20 0.34
MAPK1 P28482 1/20 0.34
RYR2 Q92736 1/20 0.34
ALDH1A1 P00352 6/20 0.33
KDM4E B2RXH2 3/20 0.33
MAPT P10636 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7070386 0.66
SCHEMBL16846586 0.66 CA1 (0.35) CA12CA1CA7CA9CA14
SCHEMBL30932111 0.66 CYP1A2 (0.38) CA12CA1CA7CA9CA14
SCHEMBL7199549 0.64 ALDH1A1 (0.33) CA12CA1CA7CA9CA14
SCHEMBL30039570 0.61 CA12 (0.43) CA12CA1CA7CA9CA14
SCHEMBL12595448 0.60
SCHEMBL2607471 0.60 DRD1 (0.62) DRD2DRD3DRD1DRD5ALDH1A1
SCHEMBL6907774 0.60 DRD1 (0.68) CA12CA1CA7CA9CA14
SCHEMBL6903663 0.60 DRD1 (0.68) CA12CA1CA7CA9CA14
SCHEMBL443070 0.60 CYP1A2 (0.79) CA12CA1CA7CA9CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0998471-B1 SUBSTITUTED HETEROCYCLIC COMPOUNDS, METHOD FOR PREPARING AND COMPOSITIONS CONTAINING SAME SERVIER LAB (FR) 2007-03-14 EP disclosed
EP-0998471-A1 SUBSTITUTED HETEROCYCLIC COMPOUNDS, METHOD FOR PREPARING AND COMPOSITIONS CONTAINING SAME ADIR ET COMPAGNIE (FR) 2000-05-10 EP disclosed
WO-1998052935-A1 SUBSTITUTED HETEROCYCLIC COMPOUNDS, METHOD FOR PREPARING AND COMPOSITIONS CONTAINING SAME ADIR ET COMPAGNIE (FR) 1998-11-26 WO disclosed