SCHEMBL5229876

SCHEMBL5229876

N#Cc1c(NC(=O)c2ccc3c(c2)OCO3)nc2c(NC=O)cccc2c1NCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 9/20 0.47
NPC1 O15118 8/20 0.47
AURKA O14965 2/20 0.45
RPS6KB1 P23443 1/20 0.45
AURKB Q96GD4 1/20 0.45
PTGS2 P35354 1/20 0.43
ALDH1A1 P00352 4/20 0.43
MAPT P10636 3/20 0.43
ALOX12 P18054 1/20 0.43
ADORA1 P30542 2/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
KDM4E B2RXH2 1/20 0.41
GAA P10253 1/20 0.41
HSD17B10 Q99714 2/20 0.41
HPGD P15428 1/20 0.41
PKM P14618 2/20 0.41
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.40
LMNA P02545 1/20 0.40
TP53 P04637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5231022 0.89 RAB9A (0.43) RAB9ANPC1AURKARPS6KB1AURKB
SCHEMBL6479836 0.87 ALDH1A1 (0.54) RAB9ANPC1AURKARPS6KB1AURKB
SCHEMBL940193 0.86 RAB9A (0.44) RAB9ANPC1AURKARPS6KB1AURKB
SCHEMBL940614 0.80 ALDH1A1 (0.44) RAB9ANPC1AURKARPS6KB1AURKB
SCHEMBL940713 0.79 RAB9A (0.43) RAB9ANPC1AURKARPS6KB1AURKB
SCHEMBL6487647 0.77 MEN1 (0.54) RAB9ANPC1PTGS2ALDH1A1MAPT
SCHEMBL940779 0.76 MAPK1 (0.45) RAB9ANPC1ALDH1A1MAPTADORA1
SCHEMBL6480798 0.73 ALDH1A1 (0.48) RAB9ANPC1ALDH1A1MAPTALOX12
SCHEMBL6489855 0.72 ADORA3 (0.49) RAB9ANPC1AURKAAURKBALDH1A1
SCHEMBL6479650 0.71 MEN1 (0.54) RAB9ANPC1ALDH1A1SMN1; SMN2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1663982-B1 AMINOQUINOLINE DERIVATIVES AND THEIR USE AS ADENOSINE A3 LIGANDS SANOFI AVENTIS (FR) 2007-11-21 EP claimed