SCHEMBL5230246

SCHEMBL5230246

ClCC=Cc1ccc(Br)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
HPGD P15428 1/20 0.42
RAB9A P51151 1/20 0.42
GRIK1 P39086 1/20 0.41
GRIK2 Q13002 1/20 0.41
CYP2A6 P11509 1/20 0.38
MEN1 O00255 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
MAPT P10636 1/20 0.37
CYP2C9 P11712 1/20 0.37
KMT2A Q03164 1/20 0.37
TUBB4A P04350 1/20 0.37
TUBB P07437 1/20 0.37
TUBA3C P0DPH7 1/20 0.37
TUBA1B P68363 1/20 0.37
TUBA4A P68366 1/20 0.37
TUBB4B P68371 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5230238 1.00 CYP2C19 (0.42) CYP2C19KDM4EALDH1A1HPGDRAB9A
SCHEMBL73285 0.78 AHR (0.50) KDM4EALDH1A1GRIK1GRIK2CYP2A6
SCHEMBL3466529 0.78 CYP2C19 (0.43) CYP2C19KDM4EALDH1A1HPGDRAB9A
SCHEMBL3466530 0.78 CYP2C19 (0.43) CYP2C19KDM4EALDH1A1HPGDRAB9A
SCHEMBL73286 0.78 AHR (0.50) KDM4EALDH1A1GRIK1GRIK2CYP2A6
SCHEMBL7631405 0.76 CYP2C19 (0.42) CYP2C19KDM4EALDH1A1HPGDRAB9A
SCHEMBL1046101 0.76 CYP2C19 (0.42) CYP2C19KDM4EALDH1A1HPGDRAB9A
SCHEMBL6397551 0.76 APP (0.52) CYP2C19KDM4EALDH1A1HPGDRAB9A
SCHEMBL256057 0.76 CYP2C19 (0.47) CYP2C19KDM4EALDH1A1HPGDRAB9A
SCHEMBL3885395 0.76 NFE2L2 (0.50) GRIK1GRIK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102241991-B Liquid crystal aligning agent, liquid crystal alignment layer manufacturing method and liquid crystal display device JSR CORP 2015-01-28 CN disclosed
CN-102241991-A Liquid crystal aligning agent, liquid crystal alignment layer manufacturing method and liquid crystal display device JSR CORP 2011-11-16 CN disclosed
EP-1737824-A2 NOVEL ALKYNE COMPOUNDS HAVING AN MCH-ANTAGONISTIC EFFECT, AND MEDICAMENTS CONTAINING SAID COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-01-03 EP disclosed
US-20050245529-A1 Alkyne compounds with MCH antagonistic activity and medicaments comprising these compounds BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2005-11-03 US disclosed
WO-2005103032-A2 NOVEL ALKYNE COMPOUNDS HAVING AN MCH-ANTAGONISTIC EFFECT, AND MEDICAMENTS CONTAINING SAID COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2005-11-03 WO disclosed
US-6831175-B2 Such as N,N-dimethyl-N-(2-((5-((E)-2-pyridin-4-ylvinyl) pyridin-3-yl)oxy)ethyl)amine ABBOTT LABORATORIES 2004-12-14 US disclosed
US-20030199511-A1 Kinase inhibitors ABBVIE INC. 2003-10-23 US disclosed
US-20030187026-A1 Kinase inhibitors ABBOTT LABORATORIES 2003-10-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030187026-A1 Kinase inhibitors MAP3K20, MAP3K19, MAP3K1 CYP2C19 2148/4885KDM4E 1738/4885ALDH1A1 3292/4885
US-20030199511-A1 Kinase inhibitors MAP3K20, MAP3K19, MAP3K1 CYP2C19 2148/4885KDM4E 1738/4885ALDH1A1 3292/4885
US-20050245529-A1 Alkyne compounds with MCH antagonistic activity and medicaments comprising these compounds MCHR1, GPR119, MCHR2 CYP2C19 3638/4885KDM4E 1952/4885ALDH1A1 3033/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.