SCHEMBL5230376

SCHEMBL5230376

NC[C@H](CO)c1ccc(F)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABBR2 O75899 5/20 0.59
GABBR1 Q9UBS5 5/20 0.59
IDO1 P14902 2/20 0.40
TDO2 P48775 2/20 0.40
AOC3 Q16853 1/20 0.40
LOXL2 Q9Y4K0 1/20 0.39
LMNA P02545 2/20 0.39
CYP2C9 P11712 2/20 0.39
CYP1A2 P05177 2/20 0.39
CYP3A4 P08684 1/20 0.39
ADORA3 P0DMS8 1/20 0.39
NFKB1 P19838 1/20 0.39
DRD3 P35462 1/20 0.39
BLM P54132 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C19 P33261 1/20 0.39
MEN1 O00255 1/20 0.39
THRB P10828 1/20 0.39
TSHR P16473 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11085032 0.86 GABBR2 (0.62) GABBR2GABBR1IDO1TDO2AOC3
SCHEMBL1772818 0.86 GABBR2 (0.47) GABBR2GABBR1IDO1TDO2AOC3
SCHEMBL5321547 0.83 GABBR2 (0.56) GABBR2GABBR1IDO1TDO2AOC3
SCHEMBL5327386 0.83 GABBR2 (0.56) GABBR2GABBR1IDO1TDO2AOC3
SCHEMBL11142937 0.80 TAAR1 (0.56) GABBR2GABBR1LMNACYP2C9CYP1A2
SCHEMBL7908792 0.78 GABBR2 (0.42) GABBR2GABBR1IDO1TDO2AOC3
SCHEMBL18595195 0.78 TRPA1 (0.42) GABBR2GABBR1AOC3LMNAMEN1
SCHEMBL9779274 0.78 GABBR2 (0.61) GABBR2GABBR1AOC3LMNACYP2C9
SCHEMBL2615282 0.78 GABBR2 (0.55) GABBR2GABBR1IDO1TDO2AOC3
SCHEMBL7396004 0.78 GABBR2 (0.61) GABBR2GABBR1AOC3LMNACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765817-A1 THIAZOLINONE UNSUBSTITUTED QUINOLINES F.HOFFMANN-LA ROCHE AG (CH) 2007-03-28 EP disclosed
WO-2006002829-A1 THIAZOLINONE UNSUBSTITUTED QUINOLINES F. HOFFMANN-LA ROCHE AG (CH) 2006-01-12 WO disclosed