SCHEMBL5230770

SCHEMBL5230770

O=C(NCc1ccc(Cl)cc1)Oc1cc(-c2ccc(O)c(F)c2)n[nH]c1=O

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.71
MAPT P10636 7/20 0.46
DAO P14920 2/20 0.41
TP53 P04637 3/20 0.41
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC10 Q969S8 1/20 0.38
HDAC11 Q96DB2 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
HDAC9 Q9UKV0 1/20 0.38
HDAC5 Q9UQL6 1/20 0.38
NCOR2 Q9Y618 1/20 0.38
ALDH2 P05091 1/20 0.37
FAAH O00519 1/20 0.36
ERCC1 P07992 1/20 0.35
ERCC4 Q92889 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5227844 0.90 GSK3B (0.57) GSK3BMAPTDAOTP53ERCC1
SCHEMBL5231030 0.89 GSK3B (0.55) GSK3BMAPTDAOTP53
SCHEMBL5231152 0.88 GSK3B (0.55) GSK3BMAPTTP53
SCHEMBL5229836 0.87 GSK3B (0.52) GSK3BMAPTDAOTP53HDAC3
SCHEMBL4855976 0.83 GSK3B (1.00) GSK3BMAPTTP53HDAC3HDAC4
SCHEMBL5234548 0.83 MAPT (0.49) GSK3BMAPTTP53
SCHEMBL5228636 0.82 GSK3B (0.48) GSK3BMAPTTP53
SCHEMBL5243212 0.79 GSK3B (0.45) GSK3BMAPTDAOTP53
SCHEMBL4848893 0.76 GSK3B (0.86) GSK3BMAPTTP53HDAC3HDAC4
SCHEMBL5235894 0.75 GSK3B (0.57) GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611121-B1 PYRIDAZINONE DERIVATIVES AS CDK2-INHIBITORS AVENTIS PHARMA SA (FR) 2007-08-08 EP claimed
EP-1581505-B1 PYRIDAZINONE DERIVATIVES AS GSK-3BETA INHIBITORS SANOFI AVENTIS DEUTSCHLAND (DE) 2007-08-01 EP claimed