SCHEMBL5227844

SCHEMBL5227844

O=C(NCc1ccc(Cl)cc1)Oc1cc(-c2ccc(O)c(Cl)c2)n[nH]c1=O

nearest known ligand 0.57

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.57
MAPT P10636 7/20 0.47
TP53 P04637 2/20 0.42
DAO P14920 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
HSD17B2 P37059 1/20 0.38
ENPP2 Q13822 1/20 0.37
ERCC1 P07992 1/20 0.37
ERCC4 Q92889 1/20 0.37
ALPL P05186 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5230770 0.90 GSK3B (0.71) GSK3BMAPTTP53DAOERCC1
SCHEMBL5231030 0.90 GSK3B (0.55) GSK3BMAPTTP53DAOALPL
SCHEMBL5231152 0.89 GSK3B (0.55) GSK3BMAPTTP53
SCHEMBL5229836 0.89 GSK3B (0.52) GSK3BMAPTTP53DAOALPL
SCHEMBL5234548 0.85 MAPT (0.49) GSK3BMAPTTP53
SCHEMBL5228636 0.84 GSK3B (0.48) GSK3BMAPTTP53ALPLMEN1
SCHEMBL4849862 0.82 GSK3B (0.81) GSK3BMAPTTP53ENPP2MEN1
SCHEMBL5243212 0.81 GSK3B (0.45) GSK3BMAPTTP53DAOMEN1
SCHEMBL5243973 0.77 TSHR (0.48) GSK3BMAPTDAO
SCHEMBL5237798 0.75 AKT3 (0.44) GSK3BMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611121-B1 PYRIDAZINONE DERIVATIVES AS CDK2-INHIBITORS AVENTIS PHARMA SA (FR) 2007-08-08 EP claimed
EP-1581505-B1 PYRIDAZINONE DERIVATIVES AS GSK-3BETA INHIBITORS SANOFI AVENTIS DEUTSCHLAND (DE) 2007-08-01 EP claimed