SCHEMBL5232235

SCHEMBL5232235

Cc1ccc(F)cc1C(=O)N1CC2CN(c3cccc(CCC(N)=O)c3)CC2C1

nearest known ligand 0.54

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 19/20 0.54
HCRTR1 O43613 18/20 0.54
CYP1A2 P05177 1/20 0.41
KCNK3 O14649 1/20 0.41
KCNK9 Q9NPC2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5237741 0.86 HCRTR1 (0.44) HCRTR2HCRTR1
SCHEMBL5231911 0.85 HCRTR1 (0.57) HCRTR2HCRTR1CYP1A2
SCHEMBL5239352 0.85 HCRTR1 (0.55) HCRTR2HCRTR1
SCHEMBL4694475 0.84 SMN1; SMN2 (0.47) CYP1A2
SCHEMBL4692413 0.84 HCRTR1 (0.53) HCRTR2HCRTR1
SCHEMBL5233538 0.83 ALDH1A1 (0.47) HCRTR2HCRTR1
SCHEMBL4694593 0.81 ALDH1A1 (0.41) HCRTR2HCRTR1
SCHEMBL5238002 0.81 HCRTR1 (0.47) HCRTR2HCRTR1
SCHEMBL5231850 0.81 HCRTR1 (0.43) HCRTR2HCRTR1
SCHEMBL5236364 0.80 HCRTR1 (0.47) HCRTR2HCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed