SCHEMBL4694593

SCHEMBL4694593

Cc1cc(C)cc(C(=O)N2CC3CN(c4cccc(CCC(N)=O)c4)CC3C2)c1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
NPSR1 Q6W5P4 1/20 0.41
PLA2G10 O15496 5/20 0.38
HCRTR1 O43613 6/20 0.37
HCRTR2 O43614 6/20 0.37
RAB9A P51151 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
HPGD P15428 1/20 0.36
KDM4E B2RXH2 1/20 0.35
HTR7 P34969 1/20 0.35
PLA2G2A P14555 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5238361 0.93 HPGD (0.43) PLA2G10RAB9ATDP1L3MBTL1HPGD
SCHEMBL5232788 0.88 CHRNB2 (0.44) PLA2G10L3MBTL1PLA2G2A
SCHEMBL5233538 0.88 ALDH1A1 (0.47) ALDH1A1NPSR1PLA2G10HCRTR1HCRTR2
SCHEMBL4692413 0.86 HCRTR1 (0.53) PLA2G10HCRTR1HCRTR2
SCHEMBL5231026 0.85 HPGD (0.42) ALDH1A1PLA2G10HPGDPLA2G2A
SCHEMBL5237823 0.85 SLC6A7 (0.36) PLA2G10HCRTR1HCRTR2HPGDPLA2G2A
SCHEMBL5237460 0.84 PLA2G10 (0.39) ALDH1A1PLA2G10HPGDHTR7PLA2G2A
SCHEMBL4694475 0.84 SMN1; SMN2 (0.47) ALDH1A1HPGD
SCHEMBL5237286 0.84 LMNA (0.43) ALDH1A1NPSR1L3MBTL1
SCHEMBL5235769 0.83 CHRNA4 (0.47) ALDH1A1PLA2G10PLA2G2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed