SCHEMBL5233198

SCHEMBL5233198

NC(=O)CCc1cccc(N2CC3CN(C(=O)c4csc5ccccc45)CC3C2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.46
LMNA P02545 1/20 0.44
HPGD P15428 1/20 0.44
HSD17B10 Q99714 3/20 0.42
CASP1 P29466 1/20 0.42
CASP7 P55210 1/20 0.42
MAPT P10636 2/20 0.41
ALDH1A1 P00352 4/20 0.41
RECQL P46063 1/20 0.41
HTR7 P34969 1/20 0.38
HCRTR1 O43613 4/20 0.38
HCRTR2 O43614 4/20 0.38
HPN P05981 1/20 0.37
ST14 Q9Y5Y6 1/20 0.37
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
HTR1A P08908 3/20 0.36
ALOX15 P16050 1/20 0.36
PDE2A O00408 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5231927 0.81 CYP2C9 (0.42) ALDH1A1HCRTR1HCRTR2CYP2C9
SCHEMBL5232788 0.81 CHRNB2 (0.44) LMNAMAPT
SCHEMBL5233812 0.80 DPP4 (0.46)
SCHEMBL5237120 0.79 HCRTR2 (0.42) HCRTR1HCRTR2ALOX15
SCHEMBL5237813 0.79 HCRTR1 (0.39) HTTMAPTALDH1A1HCRTR1HCRTR2
SCHEMBL5239352 0.79 HCRTR1 (0.55) HCRTR1HCRTR2
SCHEMBL5229090 0.78 LMNA (0.45) LMNAHCRTR1HCRTR2
SCHEMBL5231495 0.77 CHRM2 (0.39) HCRTR1HCRTR2
SCHEMBL5237460 0.77 PLA2G10 (0.39) HPGDHSD17B10ALDH1A1HTR7CYP1A2
SCHEMBL4692413 0.77 HCRTR1 (0.53) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed