SCHEMBL5233454

SCHEMBL5233454

NC(=O)C[C@@H](c1ccccc1)N1CC2CN(C(=O)c3cnc4ccccc4n3)CC2C1

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 3/20 0.49
PTK2 Q05397 1/20 0.48
HCRTR1 O43613 10/20 0.43
HCRTR2 O43614 10/20 0.43
GRM5 P41594 1/20 0.41
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
ALOX15 P16050 1/20 0.40
HSD17B10 Q99714 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5237603 0.87 TSHR (0.46) DPP4HCRTR1HCRTR2ALDH1A1
SCHEMBL5236953 0.84 DPP4 (0.50) DPP4HCRTR1HCRTR2
SCHEMBL5235073 0.83 CHRNB2 (0.53) DPP4ALDH1A1
SCHEMBL5235823 0.79 CHRM2 (0.40) HCRTR1HCRTR2
SCHEMBL4691220 0.78 DPP4 (0.50) DPP4PTK2HCRTR1HCRTR2GRM5
SCHEMBL5237860 0.77 CCL5 (0.43)
SCHEMBL5235643 0.77 CHRNB2 (0.53) ALDH1A1HPGDALOX15
SCHEMBL5237787 0.77 DPP4 (0.49) DPP4ALDH1A1HPGD
SCHEMBL5234640 0.76 HCRTR1 (0.52) HCRTR1HCRTR2ALDH1A1
SCHEMBL5232470 0.75 CCR5 (0.54) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed