SCHEMBL5234510

SCHEMBL5234510

CC(C)N(c1nn(-c2ccc(CCC3CCCCC3)cc2)cc1OC(=O)O)C(=O)[C@H]1CC[C@H](C)CC1

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.31
NAAA Q02083 1/20 0.31
MAPK11 Q15759 1/20 0.30
MAPK14 Q16539 1/20 0.30
TBK1 Q9UHD2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5228396 0.89 KMT2A (0.34)
SCHEMBL5234503 0.88 BRS3 (0.35) PARP1MAPK11MAPK14TBK1
SCHEMBL5234986 0.88 BRS3 (0.35) PARP1MAPK11MAPK14TBK1
SCHEMBL5232338 0.87 S1PR1 (0.34) PARP1
SCHEMBL5235412 0.87 NAMPT (0.31) PARP1
SCHEMBL5236797 0.84
SCHEMBL5236128 0.84 NPC1 (0.34)
SCHEMBL5233446 0.84 NPC1 (0.35)
SCHEMBL5236136 0.84
SCHEMBL5234344 0.83 ESRRA (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730116-B1 4-CARBOX PYRAZOLE DERIVATES USEFUL AS ANTI-VIRAL AGENTS SMITHKLINE BEECHAM CORP (US) 2007-09-05 EP claimed