SCHEMBL5236128

SCHEMBL5236128

Cc1ccc(-n2cc(OC(=O)O)c(N(C(=O)[C@H]3CC[C@H](C)CC3)C(C)C)n2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.34
RAB9A P51151 3/20 0.34
ADORA3 P0DMS8 1/20 0.34
ALDH1A1 P00352 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
GLA P06280 1/20 0.33
NFKB1 P19838 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
ACKR3 P25106 1/20 0.32
CA12 O43570 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA9 Q16790 1/20 0.31
KDM5B Q9UGL1 1/20 0.30
KDM4E B2RXH2 1/20 0.30
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5236797 0.92
SCHEMBL5233446 0.92 NPC1 (0.35) NPC1RAB9AADORA3ALDH1A1GLA
SCHEMBL5234344 0.91 ESRRA (0.31)
SCHEMBL5239459 0.91 KDM4E (0.33) NPC1RAB9AALDH1A1KMT2ACA12
SCHEMBL5231776 0.91 ESRRA (0.32) NPC1RAB9AALDH1A1NPSR1MEN1
SCHEMBL5232934 0.90 KDM4E (0.30) ALDH1A1KDM4E
SCHEMBL5238208 0.90 ALDH1A1 (0.38) NPC1RAB9AALDH1A1SMN1; SMN2CA12
SCHEMBL5234129 0.90 ADORA3 (0.37) ADORA3ALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL5233835 0.90 KCNJ1 (0.32) ALDH1A1SMN1; SMN2MEN1KMT2ANAMPT
SCHEMBL5229086 0.90

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730116-B1 4-CARBOX PYRAZOLE DERIVATES USEFUL AS ANTI-VIRAL AGENTS SMITHKLINE BEECHAM CORP (US) 2007-09-05 EP claimed