SCHEMBL5235906

SCHEMBL5235906

NC(=O)CCc1cccc(N2CC3CN(C(=O)c4c(Cl)cccc4Cl)CC3C2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 7/20 0.46
HCRTR2 O43614 7/20 0.46
CCR5 P51681 1/20 0.39
NPC1 O15118 1/20 0.39
GLA P06280 1/20 0.39
HPGD P15428 1/20 0.39
SLC22A12 Q96S37 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
PLA2G10 O15496 2/20 0.36
PLA2G2A P14555 2/20 0.36
HTR1A P08908 1/20 0.36
HTR2A P28223 1/20 0.36
HTR7 P34969 1/20 0.36
HTR6 P50406 1/20 0.36
CHRM1 P11229 1/20 0.35
KDM4E B2RXH2 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HSD17B10 Q99714 1/20 0.34
SLC6A7 Q99884 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4692729 0.93 HCRTR1 (0.44) HCRTR1HCRTR2
SCHEMBL5231927 0.89 CYP2C9 (0.42) HCRTR1HCRTR2
SCHEMBL5231344 0.89 HCRTR1 (0.39) HCRTR1HCRTR2CCR5SLC22A12MEN1
SCHEMBL4692413 0.87 HCRTR1 (0.53) HCRTR1HCRTR2CCR5PLA2G10
SCHEMBL5233682 0.85 HCRTR1 (0.38) HCRTR1HCRTR2SLC22A12MEN1KMT2A
SCHEMBL5232788 0.84 CHRNB2 (0.44) MEN1KMT2APLA2G10PLA2G2AHTR2A
SCHEMBL5237741 0.83 HCRTR1 (0.44) HCRTR1HCRTR2CCR5PLA2G10
SCHEMBL5236364 0.83 HCRTR1 (0.47) HCRTR1HCRTR2CCR5PLA2G10
SCHEMBL4968486 0.83 HCRTR1 (0.42) HCRTR1HCRTR2CCR5
SCHEMBL5235957 0.83 TP53 (0.40) KMT2APLA2G10PLA2G2ACHRM1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed