SCHEMBL5237688

SCHEMBL5237688

CC(C)(C)c1ccnc([AsH2])c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 3/20 0.38
ALDH1A1 P00352 5/20 0.37
HPGD P15428 1/20 0.37
ALOX15 P16050 1/20 0.37
HSD17B10 Q99714 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
PKM P14618 1/20 0.33
RECQL P46063 1/20 0.33
ADRA2A P08913 1/20 0.33
ADRA2B P18089 1/20 0.33
ADRA2C P18825 1/20 0.33
ADRA1D P25100 1/20 0.33
HTR1D P28221 1/20 0.33
HTR1B P28222 1/20 0.33
ADRA1A P35348 1/20 0.33
ADRA1B P35368 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1507293 0.77 NOS3 (0.57) KIF11ALDH1A1GAANOS3NOS2
SCHEMBL347025 0.76 CCR1 (0.48) KIF11ALDH1A1HPGDALOX15HSD17B10
SCHEMBL29373631 0.76 CCR1 (0.48) KIF11ALDH1A1HPGDALOX15HSD17B10
SCHEMBL29453375 0.76 CCR1 (0.48) KIF11ALDH1A1HPGDALOX15HSD17B10
Hydrochloric Acid SCHEMBL23538061 0.74 CCR1 (0.46) KIF11ALDH1A1HPGDALOX15HSD17B10
SCHEMBL2783812 0.74 CCR1 (0.46) KIF11ALDH1A1HPGDALOX15HSD17B10
SCHEMBL278964 0.74 LMNA (0.41) KIF11ALDH1A1HPGDALOX15HSD17B10
SCHEMBL15663789 0.74 CCR1 (0.46) KIF11ALDH1A1HPGDALOX15HSD17B10
SCHEMBL335953 0.74 CCR1 (0.46) KIF11ALDH1A1HPGDALOX15HSD17B10
SCHEMBL23459202 0.74 CCR1 (0.46) KIF11ALDH1A1HPGDALOX15HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1379505-B1 INHIBITION OF RAF KINASE USING QUINOLYL, ISOQUINOLYL OR PYRIDYL UREAS BAYER PHARMACEUTICALS CORP (US) 2007-02-28 EP disclosed
EP-1379507-A1 HETEROARYL UREAS CONTAINING NITROGEN HETERO-ATOMS AS p38 KINASE INHIBITORS Bayer Corporation (US) 2004-01-14 EP disclosed
WO-2002085859-A1 HETEROARYL UREAS CONTAINING NITROGEN HETERO-ATOMS AS p38 KINASE INHIBITORS BAYER CORPORATION (US) 2002-10-31 WO disclosed