SCHEMBL5237774

SCHEMBL5237774

O=C1CCCN1N=C(Cc1ccnc2cc(Br)ccc12)c1ccccn1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 2/20 0.35
ALK Q9UM73 1/20 0.33
SLC22A12 Q96S37 1/20 0.33
PREP P48147 1/20 0.33
ALDH1A1 P00352 3/20 0.32
GAA P10253 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
TGFBR1 P36897 1/20 0.31
NPC1 O15118 5/20 0.31
RAB9A P51151 4/20 0.31
SMN1; SMN2 Q16637 4/20 0.31
LMNA P02545 1/20 0.31
TP53 P04637 1/20 0.31
MAPK1 P28482 1/20 0.31
CYP1A2 P05177 1/20 0.31
MAPT P10636 3/20 0.31
NFKB1 P19838 2/20 0.31
NFKB2 Q00653 2/20 0.31
RELA Q04206 2/20 0.31
MEN1 O00255 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5237769 1.00 GRM5 (0.35) GRM5ALKSLC22A12PREPALDH1A1
SCHEMBL5238502 0.93 GRM5 (0.34) GRM5SLC22A12ALDH1A1GAANPSR1
SCHEMBL5238497 0.93 GRM5 (0.34) GRM5SLC22A12ALDH1A1GAANPSR1
SCHEMBL5239805 0.89 THRB (0.40) ALDH1A1GAATGFBR1SMN1; SMN2LMNA
SCHEMBL5239810 0.89 THRB (0.40) ALDH1A1GAATGFBR1SMN1; SMN2LMNA
SCHEMBL5239257 0.88 CYP1A2 (0.41) ALDH1A1NPSR1TGFBR1RAB9ASMN1; SMN2
SCHEMBL5239266 0.88 CYP1A2 (0.41) ALDH1A1NPSR1TGFBR1RAB9ASMN1; SMN2
SCHEMBL4486620 0.87 TGFBR1 (0.38) SLC22A12PREPTGFBR1
SCHEMBL8336424 0.87 TGFBR1 (0.38) SLC22A12PREPTGFBR1
SCHEMBL4486616 0.87 TGFBR1 (0.38) SLC22A12PREPTGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1397364-B1 NOVEL PYRROLE DERIVATIVES AS PHARMACEUTICAL AGENTS LILLY CO ELI (US) 2007-07-25 EP disclosed