SCHEMBL5239805

SCHEMBL5239805

O=C1CCCN1/N=C(/Cc1ccnc2cc(Cl)ccc12)c1ccccn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.40
TGFBR1 P36897 1/20 0.40
MAPK14 Q16539 1/20 0.40
PKM P14618 2/20 0.38
ALOX15 P16050 1/20 0.38
CASP1 P29466 1/20 0.38
HSD17B10 Q99714 1/20 0.38
CHKA P35790 1/20 0.38
MAPT P10636 2/20 0.37
ALDH1A1 P00352 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
LMNA P02545 1/20 0.37
GLA P06280 1/20 0.37
HPGD P15428 1/20 0.37
TSHR P16473 1/20 0.37
MAPK1 P28482 1/20 0.37
CCR5 P51681 1/20 0.37
DPP4 P27487 1/20 0.37
KDM4E B2RXH2 2/20 0.36
GAA P10253 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5239810 1.00 THRB (0.40) THRBTGFBR1MAPK14PKMALOX15
SCHEMBL5237774 0.89 GRM5 (0.35) TGFBR1MAPTALDH1A1SMN1; SMN2LMNA
SCHEMBL5237769 0.89 GRM5 (0.35) TGFBR1MAPTALDH1A1SMN1; SMN2LMNA
SCHEMBL5239257 0.88 CYP1A2 (0.41) THRBTGFBR1MAPK14HSD17B10ALDH1A1
SCHEMBL5239266 0.88 CYP1A2 (0.41) THRBTGFBR1MAPK14HSD17B10ALDH1A1
SCHEMBL5231673 0.87 THRB (0.43) THRBTGFBR1MAPK14PKMALOX15
SCHEMBL5231678 0.87 THRB (0.43) THRBTGFBR1MAPK14PKMALOX15
SCHEMBL5238643 0.86 CYP1A2 (0.38) ALDH1A1SMN1; SMN2LMNAKDM4E
SCHEMBL5238650 0.86 CYP1A2 (0.38) ALDH1A1SMN1; SMN2LMNAKDM4E
SCHEMBL5236211 0.86 GRM5 (0.37) TGFBR1HSD17B10MAPTALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1397364-B1 NOVEL PYRROLE DERIVATIVES AS PHARMACEUTICAL AGENTS LILLY CO ELI (US) 2007-07-25 EP disclosed