SCHEMBL5238712

SCHEMBL5238712

O=C(Cc1ccnc2ccccc12)c1cnccn1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.51
PLK4 O00444 1/20 0.47
CHEK1 O14757 1/20 0.47
PDPK1 O15530 1/20 0.47
PRKD3 O94806 1/20 0.47
MAP4K4 O95819 1/20 0.47
CHEK2 O96017 1/20 0.47
CDK1 P06493 1/20 0.47
PIM1 P11309 1/20 0.47
RPS6KB1 P23443 1/20 0.47
CDK2 P24941 1/20 0.47
FLT4 P35916 1/20 0.47
KDR P35968 1/20 0.47
CSNK1D P48730 1/20 0.47
CDK8 P49336 1/20 0.47
CLK2 P49760 1/20 0.47
GSK3A P49840 1/20 0.47
GSK3B P49841 1/20 0.47
IRAK1 P51617 1/20 0.47
LIMK1 P53667 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4872056 0.84 CYP1A2 (0.55) CYP1A2GSK3BLOXL2KDM4ENAPRT
SCHEMBL5236870 0.80 LOXL2 (0.45) CYP1A2PLK4CHEK1PDPK1PRKD3
SCHEMBL5238496 0.80 LOXL2 (0.45) CYP1A2PLK4CHEK1PDPK1PRKD3
SCHEMBL5233929 0.79 CYP1A2 (0.50) CYP1A2KDRLOXL2SMN1; SMN2MAPK9
SCHEMBL5238508 0.78 CYP1A2 (0.49) CYP1A2KDRLOXL2SMN1; SMN2NPC1
SCHEMBL5240712 0.78 CYP1A2 (0.49) CYP1A2LOXL2MAPK9RAB9AFAAH
SCHEMBL29987166 0.77 CYP1A2 (0.61) CYP1A2LOXL2KDM4ESMN1; SMN2CYP2C19
SCHEMBL5239658 0.77 CYP1A2 (0.61) CYP1A2LOXL2KDM4ESMN1; SMN2CYP2C19
SCHEMBL5233274 0.77 CYP1A2 (0.55) CYP1A2LOXL2KDM4ENAPRTCYP3A4
SCHEMBL5231886 0.77 MGAM (0.53) CYP1A2LOXL2KDM4ESMN1; SMN2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1397364-B1 NOVEL PYRROLE DERIVATIVES AS PHARMACEUTICAL AGENTS LILLY CO ELI (US) 2007-07-25 EP disclosed