SCHEMBL5239014

SCHEMBL5239014

CC(=O)Cc1ccc2cc(F)ccc2c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.45
AKR1C3 P42330 1/20 0.45
AKR1C2 P52895 1/20 0.45
POLB P06746 1/20 0.43
CYP1A2 P05177 2/20 0.42
SLC6A2 P23975 2/20 0.42
SLC6A3 Q01959 2/20 0.42
KDM4E B2RXH2 1/20 0.42
NPC1 O15118 1/20 0.42
LMNA P02545 1/20 0.42
TP53 P04637 1/20 0.42
CYP3A4 P08684 1/20 0.42
MAPT P10636 1/20 0.42
MAOA P21397 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
CYP2A6 P11509 1/20 0.42
CCR3 P51677 4/20 0.41
DAO P14920 1/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13942576 0.95 CYP19A1 (0.42) PTGS1AKR1C3AKR1C2POLBCYP1A2
SCHEMBL11471233 0.83 PTGS1 (0.59) PTGS1AKR1C3AKR1C2POLBCYP1A2
SCHEMBL2615110 0.82 CYP1A2 (0.64) CYP1A2SLC6A2SLC6A3KDM4ENPC1
SCHEMBL9852730 0.81 MAOB (0.55) MAOAMAOB
SCHEMBL265881 0.81 L3MBTL1 (0.56) CYP1A2SLC6A3KDM4ESMN1; SMN2CYP2A6
SCHEMBL11471175 0.81 GAA (0.51) PTGS1AKR1C3AKR1C2NPC1MAPT
SCHEMBL48545 0.80 GAA (0.53) POLBKDM4ELMNATP53CYP3A4
SCHEMBL5692811 0.79 ALOX5 (0.51) PTGS1AKR1C3AKR1C2POLBCYP1A2
SCHEMBL18537208 0.79 L3MBTL1 (0.51) PTGS1AKR1C3AKR1C2CYP1A2SLC6A3
SCHEMBL28141362 0.79 KDM4E (0.42) PTGS1AKR1C3AKR1C2POLBCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1851232-A2 DIHYDROIMIDAZOTHIAZOLE DERIVATIVES Prosidion Limited (GB) 2007-11-07 EP disclosed
WO-2006085118-A2 DIHYDROIMIDAZOTHIAZOLE DERIVATIVES PROSIDION LIMITED (GB) 2006-08-17 WO disclosed