SCHEMBL5239605

SCHEMBL5239605

CCCC(=O)C=NNc1ccc(C(=O)O)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 16/20 0.51
RAB9A P51151 15/20 0.51
NPC1 O15118 14/20 0.51
MAPT P10636 12/20 0.51
MEN1 O00255 9/20 0.48
KMT2A Q03164 9/20 0.48
SMN1; SMN2 Q16637 6/20 0.48
MITF O75030 4/20 0.48
HPGD P15428 3/20 0.48
ALDH1A1 P00352 3/20 0.48
GFER P55789 1/20 0.48
KCNH2 Q12809 1/20 0.48
ALPL P05186 1/20 0.47
MAPK1 P28482 2/20 0.47
KDM4E B2RXH2 4/20 0.46
POLB P06746 3/20 0.46
NPY1R P25929 1/20 0.46
NPY2R P49146 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
KLF5 Q13887 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10027943 0.74 NOX1 (0.47) GAARAB9ANPC1MAPTMEN1
SCHEMBL3706136 0.73 SMN1; SMN2 (0.42) GAARAB9ANPC1MAPTMEN1
SCHEMBL18731443 0.72 GAA (0.54) GAARAB9ANPC1MAPTMEN1
SCHEMBL23728221 0.71 NOX1 (0.49) GAARAB9ANPC1MAPTMEN1
SCHEMBL23728219 0.71 NOX1 (0.49) GAARAB9ANPC1MAPTMEN1
SCHEMBL265614 0.70 TP53 (0.70) RAB9ANPC1MAPTSMN1; SMN2HPGD
SCHEMBL7490760 0.70 MAPT (0.48) GAARAB9ANPC1MAPTMEN1
SCHEMBL16792666 0.70 GAA (0.48) GAARAB9ANPC1MAPTMEN1
SCHEMBL872409 0.70 HCAR3 (0.57) SMN1; SMN2MITFALDH1A1KCNH2MAPK1
SCHEMBL455156 0.69 HCAR3 (0.55) GAAMAPTKMT2ASMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761539-A1 INDOLE DERIVATIVE AND USE FOR TREATMENT OF CANCER Takeda Pharmaceutical Company Limited (JP) 2007-03-14 EP disclosed
WO-2005118587-A1 INDOLE DERIVATIVE AND USE FOR TREATMENT OF CANCER TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2005-12-15 WO disclosed