SCHEMBL5239683

SCHEMBL5239683

O=C(OC(=O)C(F)(F)F)c1ccno1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.38
KDM4E B2RXH2 1/20 0.38
KMT2A Q03164 4/20 0.37
MEN1 O00255 2/20 0.37
GAA P10253 4/20 0.36
CHRNA4 P43681 2/20 0.36
CHRNB2 P17787 1/20 0.36
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
CHRNA7 P36544 1/20 0.36
NPC1 O15118 1/20 0.35
MAPK1 P28482 1/20 0.35
GFER P55789 3/20 0.34
GPR6 P46095 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
RXFP2 Q8WXD0 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27876363 0.76 KMT2A (0.38) MAPTKDM4EKMT2AMEN1GAA
SCHEMBL4066379 0.73
SCHEMBL27814361 0.73 KMT2A (0.41) MAPTKDM4EKMT2AMEN1GAA
Trifluoroacetic Acid SCHEMBL4752538 0.72 CHRNA4 (0.41) MAPTKDM4EKMT2AMEN1GAA
Trifluoroacetic Acid SCHEMBL5239678 0.72 CHRNA4 (0.41) MAPTKDM4EKMT2AMEN1GAA
SCHEMBL27604334 0.71 KMT2A (0.50) KMT2AMEN1NPC1GFERTDP1
SCHEMBL28061402 0.71 SOAT1 (0.44) MAPTKDM4EKMT2AMEN1GAA
SCHEMBL28287255 0.70 KMT2A (0.39) MAPTKDM4EKMT2AMEN1GAA
SCHEMBL28101508 0.70 HSD17B10 (0.50) MAPTKDM4EKMT2AMEN1NPC1
SCHEMBL28093052 0.70 CES1 (0.38) NPC1MAPK1TDP1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP disclosed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO disclosed