SCHEMBL5243643

SCHEMBL5243643

FC(F)(F)Oc1ccc(CN2Cc3cc(OCc4ccccn4)cc(Cl)c3C2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.41
PRCP P42785 5/20 0.40
MMP1 P03956 1/20 0.39
MMP2 P08253 1/20 0.39
MMP3 P08254 1/20 0.39
MMP9 P14780 1/20 0.39
MMP8 P22894 1/20 0.39
MMP14 P50281 1/20 0.39
TSHR P16473 1/20 0.38
P2RY1 P47900 3/20 0.38
TNF P01375 1/20 0.38
NOD2 Q9HC29 1/20 0.38
NOD1 Q9Y239 1/20 0.38
CHRM5 P08912 1/20 0.38
RXRA P19793 1/20 0.37
GRIN1 Q05586 1/20 0.37
GRIN2B Q13224 1/20 0.37
BCHE P06276 1/20 0.37
ACHE P22303 1/20 0.37
BACE1 P56817 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2026199 0.80 CHRM5 (0.42) MMP1MMP2MMP3MMP9MMP8
SCHEMBL5243815 0.78 ALDH1A1 (0.52) ALDH1A1PRCPTSHRTNFNOD2
SCHEMBL27684984 0.78 SCN9A (0.38) ALDH1A1PRCPMMP1MMP2MMP3
SCHEMBL2024371 0.74 GRM2 (0.49) MMP1MMP2MMP3MMP9MMP8
SCHEMBL12442167 0.73 GRM2 (0.42) MMP1MMP2MMP3MMP9MMP8
SCHEMBL5243418 0.73 ALDH1A1 (0.50) ALDH1A1TSHRTNFNOD2NOD1
SCHEMBL27703936 0.72 SCN9A (0.40) ALDH1A1MMP1MMP2MMP3MMP9
SCHEMBL5239908 0.71 ALDH1A1 (0.52) ALDH1A1TSHRTNFNOD2NOD1
SCHEMBL5279985 0.71 CHRM5 (0.48) ALDH1A1TSHRCHRM5KCNH2RAB9A
SCHEMBL2023227 0.69 LSS (0.46) ALDH1A1P2RY1TNFNOD2NOD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1778634-A1 ISOINDOLONE COMPOUNDS AND THEIR USE AS METABOTROPIC GLUTAMATE RECEPTOR POTENTIATORS AstraZeneca AB (SE) 2007-05-02 EP claimed
WO-2006020879-A1 ISOINDOLONE COMPOUNDS AND THEIR USE AS METABOTROPIC GLUTAMATE RECEPTOR POTENTIATORS ASTRAZENECA AB (SE) 2006-02-23 WO claimed