SCHEMBL5244332

SCHEMBL5244332

CN(c1ccccc1)c1ncnc(Cl)c1N

nearest known ligand 0.53

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
EGFR P00533 7/20 0.53
CSF1R P07333 7/20 0.52
PDGFRB P09619 1/20 0.43
PDGFRA P16234 1/20 0.43
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5243561 0.85 EGFR (0.46) EGFRCSF1RPDGFRB
SCHEMBL5248227 0.84 EGFR (0.38) EGFRCSF1RPDGFRBMEN1KMT2A
SCHEMBL17815795 0.79 MAP4K4 (0.36) EGFRCSF1RPDGFRBKMT2A
SCHEMBL8856262 0.76 HTT (0.42) MEN1KMT2AMAPT
SCHEMBL10501817 0.75 MAPT (0.46) EGFRCSF1RPDGFRBPDGFRAMEN1
SCHEMBL5244451 0.74 MAPT (0.58) EGFRCSF1RPDGFRBPDGFRAMEN1
SCHEMBL21159117 0.72 NUDT1 (0.35) EGFRCSF1RKMT2AMAPT
SCHEMBL27732861 0.71 CSF1R (0.50) EGFRCSF1RPDGFRBPDGFRAMEN1
SCHEMBL10952100 0.70 EGFR (0.57) EGFRCSF1RPDGFRBPDGFRAMEN1
SCHEMBL3126298 0.70 EGFR (0.60) EGFRCSF1RPDGFRBPDGFRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1848506-A2 PYRIMIDINE-FUSED DIAZEPINE DERIVATIVES AND INDOLE-FUSED PTERIDINES Attenuon, LLC (US) 2007-10-31 EP disclosed
WO-2006089298-A2 PYRIMIDINE-FUSED DIAZEPINE DERIVATIVES AND INDOLE-FUSED PTERIDINES ATTENUON, LLC (US) 2006-08-24 WO disclosed