SCHEMBL5247663

SCHEMBL5247663

Cc1nn(C(C)C)c(Sc2cc(F)cc(F)c2)c1Cc1ccncc1

nearest known ligand 0.32

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 2/20 0.32
POLB P06746 1/20 0.31
CYP17A1 P05093 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP11B1 P15538 1/20 0.31
CYP11B2 P19099 1/20 0.31
FLT1 P17948 1/20 0.31
KDR P35968 1/20 0.31
MAPK13 O15264 1/20 0.30
MAPK12 P53778 1/20 0.30
MAPK11 Q15759 1/20 0.30
MAPK14 Q16539 1/20 0.30
FYN P06241 1/20 0.30
AR P10275 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5244657 0.86 FLT1 (0.37) P2RX7POLBFLT1KDR
SCHEMBL5207323 0.85 FYN (0.31) FYN
SCHEMBL5244357 0.83 AR (0.35) AR
SCHEMBL5243356 0.79 AR (0.35) FLT1KDRAR
SCHEMBL5641863 0.76 LOXL2 (0.33) P2RX7
SCHEMBL5640684 0.75 ALDH1A1 (0.38)
SCHEMBL5640690 0.74 RECQL (0.33)
SCHEMBL5645787 0.74 P2RX7 (0.35) P2RX7POLB
SCHEMBL5244652 0.74 FLT1 (0.34) FLT1KDR
SCHEMBL5640374 0.73 MEN1 (0.35) CYP17A1CYP3A4CYP11B1FLT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1401826-B1 PYRAZOLE DERIVATIVES AS HIV REVERSE TRANSCRIPTASE INHIBITORS HOFFMANN LA ROCHE (CH) 2007-03-21 EP claimed