SCHEMBL5248023

SCHEMBL5248023

CN(Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1)CC1(N2CCNCC2)Cc2ccccc2C1

nearest known ligand 0.42

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 18/20 0.42
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
MITF O75030 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4830251 0.99 TACR1 (0.41) TACR1CYP3A4CYP2D6MITF
SCHEMBL5245485 0.94 TACR1 (0.43) TACR1
Hydrochloric Acid SCHEMBL4835695 0.93 TACR1 (0.43) TACR1
SCHEMBL5250554 0.91 SLC6A4 (0.45) TACR1
Hydrochloric Acid SCHEMBL4827379 0.90 SLC6A4 (0.44) TACR1
SCHEMBL5245183 0.85 TACR1 (0.37) TACR1
Hydrochloric Acid SCHEMBL4834834 0.84 TACR1 (0.36) TACR1
SCHEMBL5249405 0.83 SIGMAR1 (0.40) CYP3A4
SCHEMBL5244849 0.83 TACR1 (0.37) TACR1CYP3A4CYP2D6
SCHEMBL5248733 0.83 TACR1 (0.37) TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1707564-B1 Indanyl-piperazine derivatives, process for their preparation and pharmaceutical compositions containing them SERVIER LAB (FR) 2007-09-12 EP disclosed
EP-1707564-A2 Indanyl-piperazine derivatives, process for their preparation and pharmaceutical compositions containing them Les Laboratoires Servier (FR) 2006-10-04 EP disclosed