SCHEMBL5248698

SCHEMBL5248698

c1cnc(C2CCc3ccccc3N2)nc1

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 3/20 0.38
ESR1 P03372 1/20 0.37
ESR2 Q92731 1/20 0.37
SMYD3 Q9H7B4 1/20 0.37
ADRA1A P35348 1/20 0.36
AR P10275 1/20 0.36
IDH1 O75874 6/20 0.35
NPC1 O15118 1/20 0.34
MAPK13 O15264 1/20 0.34
MAPK12 P53778 1/20 0.34
MAPK11 Q15759 1/20 0.34
MAPK14 Q16539 1/20 0.34
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16037063 0.83 DDB1 (0.41) MTNR1AESR1ESR2SMYD3ADRA1A
SCHEMBL29746175 0.83 DDB1 (0.41) MTNR1AESR1ESR2SMYD3ADRA1A
SCHEMBL30124970 0.77 ESR1 (0.51) MTNR1AESR1ESR2SMYD3NPC1
SCHEMBL13784817 0.77 ESR1 (0.51) MTNR1AESR1ESR2SMYD3NPC1
SCHEMBL5051433 0.77 ESR1 (0.51) MTNR1AESR1ESR2SMYD3NPC1
SCHEMBL13306192 0.77 ESR1 (0.51) MTNR1AESR1ESR2SMYD3NPC1
SCHEMBL27733428 0.76 NOS3 (0.41) MTNR1AESR1ESR2SMYD3ADRA1A
SCHEMBL16585796 0.76 CHRNB2 (0.51) GAAMAPT
Hydrochloric Acid SCHEMBL30542604 0.75 ESR1 (0.50) MTNR1AESR1ESR2SMYD3NPC1
Hydrochloric Acid SCHEMBL26613448 0.75 ESR1 (0.50) MTNR1AESR1ESR2SMYD3NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1848506-A2 PYRIMIDINE-FUSED DIAZEPINE DERIVATIVES AND INDOLE-FUSED PTERIDINES Attenuon, LLC (US) 2007-10-31 EP disclosed
WO-2006089298-A2 PYRIMIDINE-FUSED DIAZEPINE DERIVATIVES AND INDOLE-FUSED PTERIDINES ATTENUON, LLC (US) 2006-08-24 WO disclosed