SCHEMBL5249581

SCHEMBL5249581

O=C(NCC(F)(F)F)c1ccc(-n2cc(C(=O)NCc3cccc(-c4ccc(F)cc4)c3)nn2)c(OCCOCCF)c1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 2/20 0.42
PSEN2 P49810 2/20 0.42
APH1B Q8WW43 2/20 0.42
NCSTN Q92542 2/20 0.42
APH1A Q96BI3 2/20 0.42
PSENEN Q9NZ42 2/20 0.42
DDT P30046 3/20 0.39
ULK1 O75385 2/20 0.39
GLS O94925 2/20 0.38
CNR1 P21554 1/20 0.37
AURKA O14965 1/20 0.36
ROCK2 O75116 2/20 0.36
ROCK1 Q13464 2/20 0.36
IDO1 P14902 1/20 0.36
MIF P14174 1/20 0.35
BCL9 O00512 2/20 0.35
CTNNB1 P35222 2/20 0.35
EPHX2 P34913 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3111267 0.92 GLS (0.43) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL5247497 0.91 PSEN1 (0.45) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL5246077 0.91 MMP13 (0.37) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL5246041 0.89 MIF (0.45) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL5248109 0.89 EGLN1 (0.38) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL5244307 0.88 DDT (0.50) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL5250510 0.88 DDT (0.41) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL5248520 0.88 DDT (0.41) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL5244881 0.87 GLS (0.49) GLSROCK2ROCK1
SCHEMBL5247215 0.87 DDT (0.46) PSEN1PSEN2APH1BNCSTNAPH1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1867331-A1 TRIAZOLE DERIVATIVE AND THE USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2007-12-19 EP disclosed