SCHEMBL5249643

SCHEMBL5249643

Nc1nccc(Br)c1C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAPRT Q6XQN6 1/20 0.46
KDM4E B2RXH2 9/20 0.41
ALDH1A1 P00352 4/20 0.41
GABRP O00591 3/20 0.41
GABRD O14764 3/20 0.41
GABRA1 P14867 3/20 0.41
GABRB1 P18505 3/20 0.41
GABRG2 P18507 3/20 0.41
GABRB3 P28472 3/20 0.41
GABRA5 P31644 3/20 0.41
GABRA3 P34903 3/20 0.41
GABRA2 P47869 3/20 0.41
GABRB2 P47870 3/20 0.41
GABRA4 P48169 3/20 0.41
GABRE P78334 3/20 0.41
GABRA6 Q16445 3/20 0.41
GABRG1 Q8N1C3 3/20 0.41
GABRG3 Q99928 3/20 0.41
GABRQ Q9UN88 3/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19857454 0.82 NAPRT (0.57) NAPRTKDM4EALDH1A1GABRPGABRD
SCHEMBL22688908 0.79 NAPRT (0.48) NAPRTKDM4EALDH1A1GABRPGABRD
SCHEMBL27945025 0.79 KDM4E (0.44) NAPRTKDM4EALDH1A1GABRPGABRD
SCHEMBL5355271 0.78 NAPRT (0.47) NAPRTKDM4EALDH1A1GABRPGABRD
SCHEMBL517935 0.78 KDM4E (0.55) KDM4EALDH1A1GABRPGABRDGABRA1
SCHEMBL1137039 0.78 KDM4E (0.42) NAPRTKDM4EALDH1A1GABRPGABRD
SCHEMBL20520335 0.77 NAPRT (0.47) NAPRTKDM4EALDH1A1GABRPGABRD
SCHEMBL23971140 0.76 SMN1; SMN2 (0.46) NAPRTKDM4EALDH1A1SMN1; SMN2ASPH
SCHEMBL11819966 0.76 NAPRT (0.46) NAPRTKDM4EALDH1A1GABRPGABRD
SCHEMBL23830172 0.76 KDM4E (0.41) KDM4EALDH1A1SMN1; SMN2ASPHKDM8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106565684-A 6-pyrromonazole substituted quinazoline compound, and derivative, synthetic method and application thereof 南方医科大学 2017-04-19 CN claimed
CN-104592217-B 3 (1,3,4 oxadiazolyl) 5 phenoxypyridines analog derivative and preparation method and application 沈阳药科大学 2018-03-13 CN disclosed
CN-104592217-A 3-(1, 3, 4-oxadiazol)-5-phenoxy-pyridine derivative, preparation method and application thereof UNIV SHENYANG PHARMACEUTICAL 2015-05-06 CN disclosed
EP-1781654-A1 PYRROLO-PYRIDINE KINASE MODULATORS SGX Pharmaceuticals, Inc. (US) 2007-05-09 EP disclosed
WO-2006015123-A1 PYRROLO-PYRIDINE KINASE MODULATORS SGX PHARMACEUTICALS, INC. (US) 2006-02-09 WO disclosed
EP-1623216-A2 COMPOUND LIBRARIES AND METHODS FOR DRUG DISCOVERY SGX Pharmaceuticals, Inc. (US) 2006-02-08 EP disclosed
WO-2004092727-A2 COMPOUND LIBRARIES AND METHODS FOR DRUG DISCOVERY STRUCTURAL GENOMIX, INC. (US) 2004-10-28 WO disclosed