SCHEMBL5250417

SCHEMBL5250417

CC(C)(C)C1CCC(NC(=O)c2nnn(-c3ccc(C(=O)NCC(F)(F)F)cc3)c2COCc2ccccc2)CC1

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SLC6A5 Q9Y345 2/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.38
MAPK11 Q15759 1/20 0.37
MAPK14 Q16539 1/20 0.37
MAPT P10636 1/20 0.36
CHRM4 P08173 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
HPGDS O60760 2/20 0.36
GABRA5 P31644 1/20 0.35
BRD4 O60885 1/20 0.35
TTK P33981 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3113152 0.94 SLC6A5 (0.42) SLC6A5MAPK11MAPK14CHRM4MEN1
SCHEMBL5244846 0.87 SLC6A5 (0.37) SLC6A5CHRM4MEN1KMT2AHPGDS
SCHEMBL3112209 0.87 SLC6A5 (0.40) SLC6A5MAPK11MAPK14CHRM4HPGDS
Trifluoroacetic Acid SCHEMBL5247595 0.86 SLC6A5 (0.51) SLC6A5CHRM4MEN1KMT2A
SCHEMBL3118328 0.85 BRD4 (0.42) MAPK11MAPK14MAPTCHRM4BRD4
SCHEMBL5250048 0.84 EPHX2 (0.46) MAPK14MEN1KMT2A
Trifluoroacetic Acid SCHEMBL5247913 0.84 DRD2 (0.49) SLC6A5CHRM4
SCHEMBL3113582 0.83 HPGD (0.42) MEN1KMT2A
SCHEMBL3111992 0.83 SPHK2 (0.45) MEN1KMT2AGABRA5BRD4
SCHEMBL5245587 0.83 RAB9A (0.49) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1867331-A1 TRIAZOLE DERIVATIVE AND THE USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2007-12-19 EP disclosed