SCHEMBL5250433

SCHEMBL5250433

O=C(NCc1ccc(F)cc1)c1nc(C2CSCCN2C(=O)O)nc(O)c1O

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
ERCC1 P07992 1/20 0.40
FEN1 P39748 1/20 0.40
ERCC4 Q92889 1/20 0.40
KCNH2 Q12809 1/20 0.40
CYP2C9 P11712 1/20 0.40
ALDH1A1 P00352 4/20 0.39
CALCA P06881 1/20 0.39
KCNE1 P15382 1/20 0.38
CCR1 P32246 1/20 0.38
KCNQ1 P51787 1/20 0.38
HTT P42858 1/20 0.37
PTGER4 P35408 1/20 0.37
MAPT P10636 2/20 0.36
LMNA P02545 1/20 0.36
TP53 P04637 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14609943 0.93 KCNH2 (0.41) GAANPSR1ERCC1FEN1ERCC4
SCHEMBL5119878 0.92 KCNH2 (0.41) GAANPSR1ERCC1FEN1ERCC4
SCHEMBL5128506 0.89 KCNE1 (0.43) GAANPSR1ERCC1FEN1ERCC4
SCHEMBL14609899 0.88 CYP2C9 (0.42) GAANPSR1ERCC1FEN1ERCC4
SCHEMBL5128461 0.87 MEN1 (0.42) NPSR1ERCC1FEN1ERCC4KCNH2
SCHEMBL5120394 0.86 CALCA (0.41) GAANPSR1ERCC1FEN1ERCC4
SCHEMBL5115008 0.83 KCNE1 (0.44) NPSR1ERCC1FEN1ERCC4KCNH2
SCHEMBL5117833 0.81 ALDH1A1 (0.42) NPSR1ERCC1FEN1ERCC4KCNH2
SCHEMBL5250292 0.80 KCNE1 (0.41) GAANPSR1ERCC1FEN1ERCC4
SCHEMBL5114587 0.79 KCNH2 (0.42) GAANPSR1ERCC1FEN1ERCC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1441734-B1 DIHYDROXYPYRIMIDINE CARBOXAMIDE INHIBITORS OF HIV INTEGRASE ANGELETTI P IST RICHERCHE BIO (IT) 2007-02-28 EP claimed