SCHEMBL5250837

SCHEMBL5250837

O=C(NCC(F)(F)F)c1ccc(-n2nnc(C(=O)NCc3ccc4c(c3)OCO4)c2COCc2ccccc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.54
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
ALDH1A1 P00352 4/20 0.48
HSD17B10 Q99714 2/20 0.48
KDM4E B2RXH2 1/20 0.48
TSHR P16473 1/20 0.48
HPGD P15428 1/20 0.47
MAPT P10636 1/20 0.47
HSP90AA1 P07900 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
NPSR1 Q6W5P4 1/20 0.44
POLB P06746 1/20 0.44
LMNA P02545 1/20 0.44
MAPK1 P28482 1/20 0.44
MMP13 P45452 1/20 0.44
MCHR1 Q99705 1/20 0.44
NAMPT P43490 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5250048 0.89 EPHX2 (0.46) SMN1; SMN2MEN1KMT2AHPGDLMNA
SCHEMBL5249014 0.88 CCR1 (0.45) SMN1; SMN2MEN1KMT2AHPGDLMNA
SCHEMBL5248465 0.87 CCR1 (0.46) SMN1; SMN2MEN1KMT2ALMNA
SCHEMBL5245586 0.87 CCR1 (0.46) MEN1KMT2AHPGDMAPTLMNA
SCHEMBL5244893 0.86 MAPK14 (0.48) NAMPT
SCHEMBL5244539 0.86 SMO (0.44) SMN1; SMN2MEN1KMT2AHPGDMAPT
SCHEMBL5249146 0.86 CCR1 (0.51) MEN1KMT2AMAPTTDP1NPSR1
SCHEMBL5244716 0.86 CCR1 (0.57) MEN1KMT2AMAPTTDP1LMNA
SCHEMBL5247796 0.86 CCR1 (0.45) MEN1KMT2AHPGDMAPTPOLB
SCHEMBL5247431 0.86 RIPK1 (0.44) SMN1; SMN2MEN1KMT2AHPGDLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1867331-A1 TRIAZOLE DERIVATIVE AND THE USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2007-12-19 EP disclosed